Terazosin

Terazosin

SCHEMBL41545

COc1cc2nc(N3CCN(C(=O)C4CCCO4)CC3)nc(N)c2cc1OC.Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1D

The experimentally established mechanism targets of Terazosin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D known ✓ P25100 3/20 0.98
ADRA1A known ✓ P35348 3/20 0.98
ADRA1B known ✓ P35368 3/20 0.98
KDM4E B2RXH2 5/20 1.00
ALDH1A1 P00352 4/20 1.00
GLA P06280 4/20 1.00
HPGD P15428 4/20 1.00
GAA P10253 3/20 1.00
HSD17B10 Q99714 3/20 1.00
MAPK1 P28482 2/20 1.00
KMT2A Q03164 2/20 1.00
MEN1 O00255 1/20 1.00
ADRA2A P08913 2/20 0.98
ADRA2B P18089 2/20 0.98
ADRA2C P18825 2/20 0.98
DRD1 P21728 2/20 0.98
OPRM1 P35372 2/20 0.98
OPRK1 P41145 2/20 0.98
KCNH2 Q12809 2/20 0.98
TP53 P04637 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terazosin SCHEMBL5427410 1.00 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL31284920 1.00 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL5525882 1.00 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL8441173 0.99 KDM4E (0.98) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL9053035 0.99 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL5918282 0.99 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL41544 0.99 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL9195360 0.99 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL8540346 0.99 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA
Terazosin SCHEMBL3221979 0.99 KDM4E (1.00) KDM4EALDH1A1GLAHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3777 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250375376-A1 STABLE ORAL LIQUID COMPOSITION OF TERAZOSIN Novitium Pharma LLC (US) 2025-12-11 US claimed
US-12427108-B2 Stable oral liquid composition of terazosin Novitium Pharma LLC (US) 2025-09-30 US claimed
WO-2025131019-A1 COMPOSITIONS AND METHODS FOR INHIBITING EXPRESSION OF INHIBIN SUBUNIT BETA E (INHBE) SHANGHAI ARGO BIOPHARMACEUTICAL CO., LTD. (CN) 2025-06-26 WO claimed
CN-119528888-A Preparation method of small-granularity terazosin hydrochloride 迪嘉药业集团股份有限公司 2025-02-28 CN claimed
US-20240252528-A1 Methods Of Treating Metabolic Disorders And Cardiovascular Disease With Inhibin Subunit Beta E (INHBE) Inhibitors REGENERON PHARMACEUTICALS, INC. 2024-08-01 US claimed
CN-118169271-A Method for detecting alpha-adrenergic receptor blocker, SSRI and 5-ARIs and application thereof 巴中市产品质量检验检测中心 2024-06-11 CN claimed
EP-3737676-B1 ACETAL COMPOUNDS AND THERAPEUTIC USES THEREOF LIGAND PHARM INC (US) 2024-03-06 EP claimed
CN-117092227-A Method for rapidly screening multiple veterinary drug residues in milk 黑龙江飞鹤乳业有限公司 2023-11-21 CN claimed
EP-4259279-A1 METHODS OF TREATING METABOLIC DISORDERS AND CARDIOVASCULAR DISEASE WITH INHIBIN SUBUNIT BETA E (INHBE) INHIBITORS REGENERON PHARMACEUTICALS, INC. (US) 2023-10-18 EP claimed
CN-116854674-A Preparation method of terazosin hydrochloride and intermediate thereof 迪嘉药业集团股份有限公司 2023-10-10 CN claimed
EP-0708104-A1 Process and intermediate for the preparation of terazosin hydrochloride dihydrate Abbott Laboratories (US) 1996-04-24 EP claimed
US-5504207-A REACTING 4-AMINO-2-CHLORO-6,7-DIMETHOXYQUINAZOLINE WITH N-(2-TETRAHYDROFUROYL)PIPERAZINE IN ANHYDROUS POLAR SOLVENT WITHOUT ACID SCAVENGER ABBOTT LABORATORIES (US) 1996-04-02 US claimed
EP-0623612-B1 Terazosin polymorph and pharmaceutical composition ABBOTT LAB (US) 1995-11-29 EP claimed
EP-0683167-A1 Terazosin monohydrochloride and processes and intermediate for its production Abbott Laboratories (US) 1995-11-22 EP claimed
US-5412095-A Terazosin monohydrochloride and processes and intermediate for its production ABBOTT LABORATORIES (US) 1995-05-02 US claimed
EP-0623612-A1 Terazosin polymorph and pharmaceutical composition ABBOTT LABORATORIES (US) 1994-11-09 EP claimed
US-5362730-A Solvent extraction for compounds for treatment of hypertension ABBOTT LABORATORIES (US) 1994-11-08 US claimed
US-5294615-A Crystalline 1-(4-amino-6,7-dimethoxy-2-quinazolinyl)-4-(2-tetrahydrofuroyl)piperazine monohydrochloride ABBOTT LABORATORIES (US) 1994-03-15 US claimed
US-4112097-A QUINAZOLINES ABBOTT LABORATORIES (US) 1978-09-05 US claimed
US-4026894-A 2(4(TETRAHYDRO-2-FUROYL)-PIPERAZINO)-4-AMINO-6,7-DIMETHOXYQUINAZOLINE OR 2-(4(TETRAHYDROPYRAN-2-CARBONYL)-PIPERAZINYL)-4-AMINO-6,7 -DIMETHOXYQUINAZOLINE ABBOTT LABORATORIES (US) 1977-05-31 US claimed