Geldanamycin

Geldanamycin

SCHEMBL4155

COC1=C2C[C@H](C)C[C@@H](OC)[C@H](O)[C@H](C)/C=C(/C)[C@@H](OC(N)=O)[C@H](OC)/C=C\C=C(\C)C(=O)NC(=CC1=O)C2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 1.00
HSP90AA1 P07900 17/20 0.80
ERBB2 P04626 1/20 0.79
HSP90AB1 P08238 3/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Geldanamycin SCHEMBL16669998 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL14626015 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL13928050 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL14399626 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL254191 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL12671560 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL254142 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL17973297 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL14583125 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1
Geldanamycin SCHEMBL13101681 1.00 ALDH1A1 (1.00) ALDH1A1HSP90AA1ERBB2HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 32930 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4746898-A2 IDENTIFICATION OF SEQUENCE VARIANTS OF THE ERVMER34-1 SEQUENCE FAMILY AND USE IN ANTI-CANCER THERAPIES The United States of America, as represented by the Secretary, Department of Health and Human Services (US) 2026-05-27 EP claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
EP-3841097-B1 2,6-BIS(((1H-BENZO[D]IMIDAZOL-2-YL)THIO)METHYL)PYRIDINE AND N2,N6-DIBENZYLPYRIDINE-2,6-DICARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITORS FOR TREATING CANCER BIOMEDICAL RES FOUNDATION OF THE ACADEMY OF ATHENS BRFAA (GR) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
EP-4739678-A2 AGE-MODULATING COMPOUNDS AND METHODS FOR MAKING AGE-MODULATED CELLS Memorial Sloan Kettering Cancer Center (US) 2026-05-13 EP claimed
US-20260125647-A1 AGE-MODULATING COMPOUNDS AND METHODS FOR MAKING AGE-MODULATED CELLS MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2026-05-07 US claimed
US-20260108476-A1 2,4 DNP and Prodrugs Thereof for Treatment of Cancer MITOCHON PHARMACEUTICALS, INC. (US) 2026-04-23 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-4727558-A1 NOVEL METHOD EMPLOYING ANTIBIOTICS WITH ACCRETION TO APATITE COATED IMPLANTS PREVENTING BACTERIAL ATTACHMENT AND INFECTION Moroxite I AB (SE) 2026-04-22 EP claimed
EP-4729525-A1 NEWLY SYNTHESIZED BORON-NITROGEN HETEROCYCLES AND THEIR CONJUGATES WITH PHARMACEUTICALLY UTILIZABLE SUBSTANCES Julius-Maximilians-Universität Würzburg (DE) 2026-04-22 EP claimed
WO-1999021552-A1 USE OF NON-IMMUNOSUPPRESSIVE COMPOUNDS FOR PROMOTING NERVE REGENERATION OREGON HEALTH SCIENCES UNIVERSITY (US) 1999-05-06 WO claimed
WO-1998051702-A1 METHODS AND COMPOSITIONS FOR DESTRUCTION OF SELECTED PROTEINS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1998-11-19 WO claimed
CN-1189340-A Novel grand spectrum anti-virus application of Gerd mycomycin TAO PEIZHEN (CN) 1998-08-05 CN claimed
WO-1998029110-A2 FORMULATION AND METHOD FOR TREATING NEOPLASMS BY INHALATION BATTELLE MEMORIAL INSTITUTE (US) 1998-07-09 WO claimed
EP-0828418-A1 INDUCEMENT OF THERMOTOLERANCE WITH BENZOQUINONOID ANSAMYCINS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-03-18 EP claimed
US-5626757-A RESOLUTION OF ENANTIOMORPHS BY ELECTROPHORESIS AND CHROMATOGRAPHY ADVANCED SEPARATION TECHNOLOGIES INC. (US) 1997-05-06 US claimed
WO-1996034525-A1 INDUCEMENT OF THERMOTOLERANCE WITH BENZOQUINONOID ANSAMYCINS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1996-11-07 WO claimed
EP-0664702-A1 TUMORICIDAL ACTIVITY OF BENZOQUINONOID ANSAMYCINS AGAINST PROSTATE CANCER AND PRIMITIVE NEURAL MALIGNANCIES THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-08-02 EP claimed
WO-1994008578-A2 TUMORICIDAL ACTIVITY OF BENZOQUINONOID ANSAMYCINS AGAINST PROSTATE CANCER AND PRIMITIVE NEURAL MALIGNANCIES THE GOVERNMENT OF THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1994-04-28 WO claimed
US-4261989-A Geldanamycin derivatives and antitumor drug KAKEN CHEMICAL CO. LTD. (JP) 1981-04-14 US claimed