SCHEMBL4155314

SCHEMBL4155314

NC(=O)c1cccc(-c2cncc(NCc3cccc(Cl)c3)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 3/20 0.55
RPS6KB1 P23443 3/20 0.47
AKT1 P31749 1/20 0.47
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
NPC1 O15118 1/20 0.46
CLK1 P49759 1/20 0.46
FYN P06241 2/20 0.46
PARP1 P09874 1/20 0.46
ADRB2 P07550 1/20 0.44
ADRB1 P08588 1/20 0.44
ADRB3 P13945 1/20 0.44
CD38 P28907 1/20 0.43
MAPT P10636 1/20 0.43
THRB P10828 1/20 0.43
CYP11B2 P19099 1/20 0.43
SCN2A Q99250 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4153724 0.90 MAP4K4 (0.49) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4155753 0.88 S1PR1 (0.46) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4143243 0.88 FYN (0.57) VNN1RPS6KB1CLK1FYNPARP1
SCHEMBL4156327 0.86 CLK1 (0.50) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4190030 0.85 FYN (0.60) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4143026 0.85 MKNK1 (0.50) VNN1RPS6KB1HDAC1CLK1FYN
SCHEMBL4140370 0.85 CLK1 (0.48) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4155055 0.84 FYN (0.53) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4140030 0.84 FYN (0.53) VNN1RPS6KB1HDAC1HDAC6CLK1
SCHEMBL4191971 0.82 HDAC1 (0.47) HDAC1HDAC2CLK1FYNMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090163515-A1 Compounds Which Bind to the Active Site of Protein Kinase Enzymes BIOFOCUS DISCOVERY LTD. 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163515-A1 Compounds Which Bind to the Active Site of Protein Kinase Enzymes ROCK1, ROCK2, CIT VNN1 4724/4885RPS6KB1 736/4885AKT1 83/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.