SCHEMBL4157040

SCHEMBL4157040

O=C(O)c1cccc(NC(=O)c2ccc3nc(-c4c(Cl)cccc4Cl)[nH]c3c2)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.75
NR2E3 Q9Y5X4 2/20 0.56
MMP2 P08253 1/20 0.53
MMP9 P14780 1/20 0.53
COMT P21964 1/20 0.53
MMP8 P22894 1/20 0.53
MMP13 P45452 1/20 0.53
CHEK2 O96017 2/20 0.53
PRSS12 P56730 1/20 0.52
KDM4E B2RXH2 1/20 0.51
MEN1 O00255 1/20 0.51
NPC1 O15118 1/20 0.51
POLB P06746 1/20 0.51
MAPT P10636 1/20 0.51
THRB P10828 1/20 0.51
RECQL P46063 1/20 0.51
RAB9A P51151 1/20 0.51
KMT2A Q03164 1/20 0.51
ATM Q13315 1/20 0.51
KDR P35968 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1250343 0.95 DGAT1 (0.80) DGAT1NR2E3MMP2MMP9COMT
SCHEMBL1250241 0.92 DGAT1 (0.75) DGAT1NR2E3MMP2MMP9COMT
SCHEMBL1249930 0.91 DGAT1 (0.85) DGAT1NR2E3MMP2MMP9COMT
SCHEMBL1249424 0.89 DGAT1 (0.82) DGAT1NR2E3CHEK2KDM4EMEN1
SCHEMBL1251151 0.89 DGAT1 (0.71) DGAT1NR2E3COMTMEN1NPC1
SCHEMBL1248424 0.88 DGAT1 (0.67) DGAT1MMP2MMP9MMP8MMP13
SCHEMBL1250402 0.87 DGAT1 (0.75) DGAT1NR2E3MMP2MMP9MMP8
SCHEMBL1249997 0.87 DGAT1 (0.82) DGAT1NR2E3CHEK2KDM4EMEN1
SCHEMBL1250221 0.87 DGAT1 (0.85) DGAT1NR2E3CHEK2KDRITGB1
SCHEMBL11411628 0.86 DGAT1 (0.68) DGAT1NR2E3CHEK2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074089-A2 ORGANIC COMPOUNDS Novartis AG (CH) 2009-07-01 EP disclosed
WO-2008048991-A2 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2008-04-24 WO disclosed