SCHEMBL4159372

SCHEMBL4159372

COCc1nc2c(N)nc3cccnc3c2n1CCN

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 11/20 0.47
TLR7 Q9NYK1 11/20 0.43
NUDT1 P36639 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.37
PRMT5 O14744 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALOX12 P18054 1/20 0.37
HTT P42858 1/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4160877 0.89 TLR7 (0.46) TLR8TLR7
Hydrochloric Acid SCHEMBL4152038 0.88 TLR7 (0.46) TLR8TLR7
SCHEMBL20474545 0.83 TLR8 (0.38) TLR8TLR7NUDT1KDM4ENPC1
SCHEMBL4147486 0.83 TLR7 (0.52) TLR8TLR7NUDT1HTT
SCHEMBL3350352 0.83 TLR7 (0.63) TLR8TLR7
SCHEMBL4160522 0.81 TLR7 (0.56) TLR8TLR7
SCHEMBL4157089 0.80 TLR7 (0.49) TLR8TLR7NUDT1L3MBTL1KDM4E
SCHEMBL4383648 0.79 PRMT5 (0.38) TLR8TLR7PRMT5
SCHEMBL2749012 0.79 TLR8 (0.55) TLR8TLR7NUDT1
SCHEMBL28765453 0.77 TLR8 (0.53) TLR8TLR7NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8846710-B2 Method of preferentially inducing the biosynthesis of interferon 3M INNOVATIVE PROPERTIES COMPANY (US) 2014-09-30 US disclosed
US-8343993-B2 Hydroxyalkyl substituted imidazonaphthyridines 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-01-01 US disclosed
US-20090253695-A1 Hydroxyalkyl Substituted Imidazonaphthyridines COLEY PHARMACEUTICAL GROUP, INC, (US) 2009-10-08 US disclosed
US-20090030031-A1 Method of Preferentially Inducing the Biosynthesis of Interferon COLEY PHARMACEUTICAL GROUP, INC. (US) 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090030031-A1 Method of Preferentially Inducing the Biosynthesis of Interferon IFNG, IFNAR1, EIF2AK2 TLR8 494/4885TLR7 194/4885NUDT1 302/4885
US-20090253695-A1 Hydroxyalkyl Substituted Imidazonaphthyridines IFNG, IFNAR1, IRF3 TLR8 187/4885TLR7 68/4885NUDT1 148/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.