Fluvastatin

Fluvastatin

SCHEMBL41662

CC(C)n1c(/C=C/[C@@H](O)C[C@@H](O)CC(=O)O)c(-c2ccc(F)cc2)c2ccccc21.[NaH]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HMGCR

The experimentally established mechanism targets of Fluvastatin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR known ✓ P04035 7/20 0.98
CYP2C9 P11712 4/20 0.98
SIRT6 Q8N6T7 2/20 0.98
NR4A2 P43354 2/20 0.98
PDE4D Q08499 2/20 0.98
TBXA2R P21731 2/20 0.98
ADRA1A P35348 2/20 0.98
ABCC3 O15438 1/20 0.98
ABCB11 O95342 1/20 0.98
PGR P06401 1/20 0.98
ADORA3 P0DMS8 1/20 0.98
RXRA P19793 1/20 0.98
CCKAR P32238 1/20 0.98
PTGS2 P35354 1/20 0.98
SLC10A1 Q14973 1/20 0.98
KDM4E B2RXH2 1/20 0.83
ALDH1A1 P00352 1/20 0.83
LMNA P02545 1/20 0.83
CYP1A2 P05177 1/20 0.83
SMN1; SMN2 Q16637 1/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluvastatin SCHEMBL1147657 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL6250394 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL4620256 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL1147653 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL41664 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL5072556 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL344982 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL6270543 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL246750 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D
Fluvastatin SCHEMBL28166565 1.00 HMGCR (0.98) HMGCRCYP2C9SIRT6NR4A2PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3649 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119951592-A Preparation method of catalytic material for photocatalytic degradation of carbamazepine in sewage 北方工业大学 2025-05-09 CN claimed
US-20250144067-A1 PERSONALIZED STARVATION THERAPY FOR CANCER FAETH THERAPEUTICS, INC. 2025-05-08 US claimed
CN-119185228-A Fluvastatin sodium sustained release tablet and preparation method thereof 杭州泓友医药科技有限公司 2024-12-27 CN claimed
CN-221999480-U Purification device is used in fluvastatin sodium tablet production 广州誉东健康制药有限公司 2024-11-15 CN claimed
EP-4445959-A2 PHARMACEUTICAL FORMULATIONS OF STATINS AND OMEGA-3 FATTY ACIDS FOR ENCAPSULATION Catalent Ontario Limited (CA) 2024-10-16 EP claimed
EP-3581173-B1 PHARMACEUTICAL FORMULATIONS OF STATINS AND OMEGA-3 FATTY ACIDS FOR ENCAPSULATION CATALENT ONTARIO LTD (CA) 2024-08-28 EP claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
CN-117860696-A Fluvastatin sodium sustained release preparation and preparation method thereof 浙江高跖医药科技股份有限公司 2024-04-12 CN claimed
CN-116924962-A Preparation method of fluvastatin sodium impurity F 广州瑞尔医药科技有限公司 2023-10-24 CN claimed
EP-4218765-A2 PHARMACEUTICAL COMPOSITION AND THERAPEUTIC COMBINATION COMPRISING A CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITOR AND HMG COA REDUCTASE INHIBITORS NewAmsterdam Pharma B.V. (NL) 2023-08-02 EP claimed
WO-2001056547-A2 PREPARATION OF AQUEOUS CLEAR SOLUTION DOSAGE FORMS WITH BILE ACIDS YOO SEO HONG (US) 2001-08-09 WO claimed
US-6124340-A FLUVASTATIN SODIUM FOR THE TREATMENT OF A CARDIOVASCULAR DISEASE ASTRA AKTIEBOLAG (SE) 2000-09-26 US claimed
EP-0547000-B1 Stabilized pharmaceutical compositions comprising an HMG-CoA reductase inhibitor compound NOVARTIS AG (CH) 2000-02-02 EP claimed
EP-0907639-A1 POLYMORPHIC COMPOUNDS Astra Aktiebolag (publ) (SE) 1999-04-14 EP claimed
CN-1041794-C Stabilized pharmaceutical compositions comprising an HMG-conreductase inhibitor compound SANDOZ LTD (CH) 1999-01-27 CN claimed
WO-1997049681-A1 POLYMORPHIC COMPOUNDS ASTRA AKTIEBOLAG (PUBL) (SE) 1997-12-31 WO claimed
WO-1997026874-A1 USE OF FLUVASTATIN DERIVATIVES IN SKIN DISEASE AND TOPICAL COMPOSITIONS CONTAINING THEM NOVARTIS AG (CH) 1997-07-31 WO claimed
US-5356896-A Alkaline stabiling medium SANDOZ LTD. (CH) 1994-10-18 US claimed
CN-1091634-A The stable pharmaceutical composition that contains a kind of β-Qiang Ji-β-Jia Jiwuersuandanxian coenzyme reductase inhibitor SANDOZ LTD (CH) 1994-09-07 CN claimed
EP-0547000-A1 Stabilized pharmaceutical compositions comprising an HMG-CoA reductase inhibitor compound SANDOZ LTD. (CH) 1993-06-16 EP claimed