SCHEMBL4170667

SCHEMBL4170667

CC[C@H](C)n1c(=O)[nH]c2nc(-c3cnn(Cc4cccc(C(F)(F)F)c4)c3)n(C)c2c1=O

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 19/20 0.57
ADORA2A P29274 14/20 0.57
ADORA3 P0DMS8 12/20 0.57
ADORA1 P30542 13/20 0.53
PLK4 O00444 1/20 0.49
CDK2 P24941 1/20 0.49
IRAK1 P51617 1/20 0.49
RPS6KA3 P51812 1/20 0.49
PLK3 Q9H4B4 1/20 0.49
CSNK1G3 Q9Y6M4 1/20 0.49
ALK Q9UM73 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5147140 0.82 ADORA2B (0.71) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1947236 0.78 ADORA2B (0.79) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1944491 0.76 ADORA2B (0.71) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1944916 0.75 ADORA2B (0.82) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1724513 0.74 ADORA2B (0.55) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1446900 0.73 ADORA2B (0.70) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1697135 0.73 ADORA2B (0.64) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1724705 0.73 ADORA2B (0.58) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL242942 0.73 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1945825 0.72 ADORA2B (1.00) ADORA2BADORA2AADORA3ADORA1PLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009088518-A1 A2B ADENOSINE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF CANCER CV THERAPEUTICS, INC. (US) 2009-07-16 WO disclosed