SCHEMBL4171114

SCHEMBL4171114

C=CC(=O)C(C=Cc1ccccc1)=CC#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.46
LMNA P02545 4/20 0.46
ALDH1A1 P00352 3/20 0.46
HDAC3 O15379 2/20 0.46
HDAC4 P56524 2/20 0.46
HDAC1 Q13547 2/20 0.46
HDAC2 Q92769 2/20 0.46
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
PLIN1 O60240 2/20 0.46
RECQL P46063 2/20 0.46
PLIN5 Q00G26 2/20 0.46
ABHD5 Q8WTS1 2/20 0.46
F3 P13726 2/20 0.46
TNKS O95271 1/20 0.46
HCAR2 Q8TDS4 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
TNKS2 Q9H2K2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24603 0.79 MAPT (0.50) MAPTLMNAALDH1A1HDAC3HDAC4
SCHEMBL2474967 0.76 MAPT (0.59) MAPTLMNAALDH1A1HDAC3HDAC4
Acrylonitrile SCHEMBL2549054 0.76 MAPT (0.60) MAPTLMNAALDH1A1HDAC3HDAC4
SCHEMBL2549053 0.75 MCL1 (0.41) MAPTLMNAALDH1A1HDAC3HDAC4
SCHEMBL7638028 0.74 MAPT (0.47) MAPTLMNAALDH1A1HDAC3HDAC4
SCHEMBL5608238 0.74 MAPT (0.44) MAPTLMNAALDH1A1HDAC3HDAC4
Acrylonitrile SCHEMBL28051655 0.74 HDAC3 (0.49) MAPTLMNAALDH1A1HDAC3HDAC4
SCHEMBL11870197 0.73 MAPT (0.39) MAPTLMNAALDH1A1HDAC3HDAC4
SCHEMBL295030 0.73 GLA (0.49) MAPTLMNAALDH1A1HDAC3HDAC4
Bicarbonate SCHEMBL278424 0.73 MAPT (0.43) MAPTLMNAALDH1A1HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 81 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4301810-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING ORGANIC MATERIALS, STABILIZER COMPOSITION, MASTER BATCH, COMPOSITION, MOLDING COMPOUND FOR MOLDINGS, PROCESS FOR OXIDATIVE, THERMAL AND ACTINIC STABILIZATION OF A THERMOPLASTIC, AND USE OF A COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-10 EP claimed
EP-4301809-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE RECYCLED THERMOPLASTICS, AND USE OF COMPOSITIONS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-10 EP claimed
WO-2024002875-A1 USE OF A STABILIZER COMPOSITION FOR STABILIZING HALOGEN-FREE VIRGIN THERMOPLASTICS, STABILIZER COMPOSITION, MASTER BATCH OR CONCENTRATE, STABILIZED PLASTIC COMPOSITION, PROCESS FOR STABILIZING HALOGEN-FREE VIRGIN THERMOPLASTICS, AND USE OF COMPOSITION Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-04 WO claimed
EP-4237484-A1 USE OF EUGENOL DERIVATIVES AS STABILIZERS, ORGANIC MATERIAL AND EUGENOL DERIVATIVES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-09-06 EP claimed
EP-4217200-A1 COMPOSITE COMPONENT Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-08-02 EP claimed
EP-4214275-A1 USE OF DIEUGENOL, OLIGOMERS AND/OR POLYMERS OF EUGENOL FOR STABILIZING ORGANIC MATERIALS, STABILIZED PLASTICS COMPOSITION, STABILIZER COMPOSITION AND METHOD FOR STABILIZING ORGANIC MATERIALS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-07-26 EP claimed
EP-4126810-A1 USE OF SUBSTITUTED CINNAMIC ACID ESTERS AS STABILISERS FOR ORGANIC MATERIALS, STABILISED ORGANIC MATERIAL, METHOD FOR STABILISING ORGANIC MATERIALS AND SPECIFIC CINAMIC ACID ESTERS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2023-02-08 EP claimed
WO-2022090566-A1 USE OF EUGENOL DERIVATIVES AS STABILIZERS, ORGANIC MATERIAL AND EUGENOL DERIVATIVES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-05-05 WO claimed
WO-2022058371-A1 USE OF DIEUGENOL, OLIGOMERS AND/OR POLYMERS OF EUGENOL FOR STABILIZING ORGANIC MATERIALS, STABILIZED PLASTICS COMPOSITION, STABILIZER COMPOSITION AND METHOD FOR STABILIZING ORGANIC MATERIALS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-03-24 WO claimed
EP-3947540-A1 METHOD FOR STABILIZING THERMOPLASTIC RECYCLATES, STABILIZED PLASTIC COMPOSITIONS, AND MOLDING COMPOUNDS AND MOLDED PARTS PRODUCED THEREFROM FRAUNHOFER-GESELLSCHAFT zur Förderung der angewandten Forschung e.V. (DE) 2022-02-09 EP claimed
WO-2019063550-A1 METHOD FOR STABILIZING HALOGEN-FREE THERMOPLASTIC RECYCLATES, STABILIZED PLASTIC COMPOSITIONS, AND MOLDING COMPOUNDS AND MOLDED PARTS PRODUCED THEREFROM Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2019-04-04 WO claimed
WO-2019020699-A1 HALOGEN-FREE SULPHONIC ACID ESTER AND/OR SULPHINIC ACID ESTER AS FLAME RETARDANT, FLAME RETARDANT SYNERGISTS AND RADICAL GENERATORS IN PLASTICS Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2019-01-31 WO claimed
EP-2978804-B1 USE OF ORGANIC OXY IMIDES AS FLAME RETARDANTS FOR PLASTICS AND FLAME-RETARDANT PLASTICS COMPOSITION AND MOULDINGS PRODUCED THEREFROM FRAUNHOFER GES FORSCHUNG (DE) 2018-11-07 EP claimed
WO-2018153747-A1 EFFICIENT PHOSPHOROUS STABILISERS BASED ON DIPHENYLAMINE AND HETEROCYCLIC DIPHENYLAMINE DERIVATIVES Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2018-08-30 WO claimed
EP-3194487-A1 USE OF ORGANIC OXYIMIDES AS RADICAL GENERATORS IN PLASTICS, METHOD FOR GENERATING RADICALS IN PLASTICS AND USE OF SAID METHOD Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2017-07-26 EP claimed
WO-2016042038-A1 USE OF ORGANIC OXYIMIDES AS RADICAL GENERATORS IN PLASTICS, METHOD FOR GENERATING RADICALS IN PLASTICS AND USE OF SAID METHOD Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2016-03-24 WO claimed
EP-2978804-A1 USE OF ORGANIC OXY IMIDES AS FLAME RETARDANTS FOR PLASTICS AND FLAME-RETARDANT PLASTICS COMPOSITION AND MOULDINGS PRODUCED THEREFROM Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2016-02-03 EP claimed
WO-2014154636-A1 USE OF ORGANIC OXY IMIDES AS FLAME RETARDANTS FOR PLASTICS AND FLAME-RETARDANT PLASTICS COMPOSITION AND MOULDINGS PRODUCED THEREFROM Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2014-10-02 WO claimed
WO-2014090936-A1 SYNERGISTIC COMPOSITION AND USE THEREOF AS A FLAME RETARDANT ZYLUM BETEILIGUNGSGESELLSCHAFT MBH & CO. PATENTE II KG (DE) 2014-06-19 WO claimed
EP-2743299-A1 Synergistic compound and its use as flame retardant Zylum Beteiligungsgesellschaft mbH & Co. Patente II KG (DE) 2014-06-18 EP claimed