SCHEMBL4173005

SCHEMBL4173005

c1cnc2c(c1)CC[C@@H]1CCCN(Cc3nc4ccccc4[nH]3)[C@H]21

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 17/20 0.48
DRD4 P21917 3/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 2/20 0.47
CHRM2 P08172 1/20 0.47
DRD2 P14416 1/20 0.47
OPRM1 P35372 1/20 0.47
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4173009 1.00 CXCR4 (0.48) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL13875192 1.00 CXCR4 (0.48) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL4182113 1.00 CXCR4 (0.48) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL13875273 0.94 DRD4 (0.48) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL4178914 0.94 DRD4 (0.48) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL4175818 0.84 DRD4 (0.43) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL13875275 0.84 DRD4 (0.43) CXCR4DRD4CYP3A4CYP2D6CHRM2
SCHEMBL13875216 0.81 CXCR4 (0.60) CXCR4DRD4CYP2D6KCNH2
SCHEMBL4170853 0.81 CXCR4 (0.60) CXCR4DRD4CYP2D6KCNH2
SCHEMBL5548249 0.81 CXCR4 (0.60) CXCR4DRD4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090093454-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2009-04-09 US disclosed
US-20090093454-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2009-04-09 US disclosed
US-20090093454-A1 Chemical Compounds SMITHKLINE BEECHAM CORPORATION 2009-04-09 US disclosed
EP-1853604-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2007-11-14 EP disclosed
WO-2006096444-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090093454-A1 Chemical Compounds SLC10A1, CYP11B2, CYP4F3 CXCR4 2681/4885DRD4 1190/4885CYP3A4 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.