SCHEMBL4176541

SCHEMBL4176541

CCCCN(CCCC)c1ccc(C2=CC(=O)C(=O)c3ccccc32)cc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 11/20 0.55
PTPRC P08575 5/20 0.54
PTPRF P10586 2/20 0.54
CDC25B P30305 2/20 0.54
APAF1 O14727 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
AR P10275 1/20 0.40
CNR2 P34972 1/20 0.40
MALT1 Q9UDY8 1/20 0.40
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4192820 0.86 PTPN1 (0.61) PTPN1PTPRCPTPRFCDC25BALDH1A1
SCHEMBL4192812 0.82 PTPN1 (0.54) PTPN1PTPRCPTPRFCDC25BAPAF1
SCHEMBL1409019 0.82 PTPN1 (0.54) PTPN1PTPRCPTPRFCDC25BALDH1A1
SCHEMBL7487467 0.78 PTPN1 (0.67) PTPN1PTPRCPTPRFCDC25BCES2
SCHEMBL1772040 0.77 KDM4E (0.49) ALDH1A1ARCNR2BACE1
SCHEMBL28460266 0.75 AR (0.59) ALDH1A1ARCNR2
SCHEMBL6688709 0.74 BACE1 (0.60) PTPN1PTPRCPTPRFCDC25BALDH1A1
SCHEMBL18984697 0.74 MAPK1 (0.51) PTPRCALDH1A1ARCNR2
SCHEMBL27952438 0.73 AR (0.43) ALDH1A1ARCNR2
SCHEMBL3905368 0.72 AR (0.51) ALDH1A1ARCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090043116-A1 HETERO-POLYCYCLIC COMPOUNDS, AND COLORING MATTERS, PIGMENTS, DYES, COLOR-CHANGING MATERIAL COMPOSITIONS, AND COLOR-CHANGING FILMS, MADE BY USING THE COMPOUNDS IDEMITSU KOSAN CO., LTD. (JP) 2009-02-12 US disclosed
US-20080290329-A1 HETERO-POLYCYCLIC COMPOUNDS, AND COLORING MATTERS, PIGMENTS, DYES, COLOR-CHANGING MATERIAL COMPOSITIONS, AND COLOR-CHANGING FILMS, MADE BY USING THE COMPOUNDS IDEMITSU KOSAN CO., LTD. (JP) 2008-11-27 US disclosed
US-7420065-B2 Color-changing performance does not deteriorate even after used for long time and which is prevented from being unusable due to deposition of the coloring matter during storage IDEMITSU KOSAN CO., LTD. (JP) 2008-09-02 US disclosed
US-20060235060-A1 Hetero-polycyclic compounds, and coloring matters, pigments, dyes, color-changing material compositions, and color-changing films, made by using the compounds IDEMITSU KOSAN CO., LTD. (JP) 2006-10-19 US disclosed
EP-1593675-A1 HETERO-POLYCYCLIC COMPOUNDS, AND COLORING MATTERS, PIGMENTS, DYES, COLOR-CHANGING MATERIAL COMPOSITIONS, AND COLOR-CHANGING FILMS, MADE BY USING THE COMPOUNDS IDEMITSU KOSAN CO., LTD. (JP) 2005-11-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080290329-A1 HETERO-POLYCYCLIC COMPOUNDS, AND COLORING MATTERS, PIGMENTS, DYES, COLOR-CHANGING MATERIAL COMPOSITIONS, AND COLOR-CHANGING FILMS, MADE BY USING THE COMPOUNDS PBRM1, BICRA, PARG PTPN1 3776/4885PTPRC 2882/4885PTPRF 4202/4885
US-20090043116-A1 HETERO-POLYCYCLIC COMPOUNDS, AND COLORING MATTERS, PIGMENTS, DYES, COLOR-CHANGING MATERIAL COMPOSITIONS, AND COLOR-CHANGING FILMS, MADE BY USING THE COMPOUNDS PBRM1, BICRA, PARG PTPN1 3776/4885PTPRC 2882/4885PTPRF 4202/4885
US-20060235060-A1 Hetero-polycyclic compounds, and coloring matters, pigments, dyes, color-changing material compositions, and color-changing films, made by using the compounds PBRM1, BICRA, PARG PTPN1 3776/4885PTPRC 2882/4885PTPRF 4202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.