SCHEMBL4179745

SCHEMBL4179745

Fc1cccc(Cn2cnnc2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.65
CYP11B2 P19099 1/20 0.65
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
KDM4C Q9H3R0 1/20 0.47
HSD17B10 Q99714 1/20 0.46
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
IDO1 P14902 4/20 0.45
POLB P06746 1/20 0.45
DBH P09172 1/20 0.45
GRM2 Q14416 1/20 0.44
AGXT P21549 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3260891 0.80 NPC1 (0.71) CYP11B1CYP11B2NPC1RAB9AALDH1A1
SCHEMBL24845216 0.79 CYP11B1 (0.58) CYP11B1CYP11B2NPC1RAB9AALDH1A1
SCHEMBL9747422 0.79 CYP11B1 (1.00) CYP11B1CYP11B2POLB
SCHEMBL3383923 0.77 CYP11B1 (0.65) CYP11B1CYP11B2
SCHEMBL16129815 0.77 CYP11B1 (0.65) CYP11B1CYP11B2SMN1; SMN2TAAR1IDO1
SCHEMBL25583831 0.76 CYP11B1 (0.55) CYP11B1CYP11B2NPC1RAB9AALDH1A1
SCHEMBL2979521 0.76 CYP11B1 (0.55) CYP11B1CYP11B2NPC1RAB9AALDH1A1
SCHEMBL24845219 0.76 CYP11B1 (0.55) CYP11B1CYP11B2NPC1RAB9AALDH1A1
SCHEMBL27999080 0.76 GABRG2 (0.43) CYP11B1CYP11B2NPC1RAB9APOLB
SCHEMBL28174118 0.75 CYP19A1 (0.60) CYP11B1CYP11B2NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009095394-A1 DIAZEPANES AS HISTAMINE H3 RECEPTOR ANTAGONISTS EVOTEC NEUROSCIENCES GMBH (DE) 2009-08-06 WO disclosed
WO-2009095394-A1 DIAZEPANES AS HISTAMINE H3 RECEPTOR ANTAGONISTS EVOTEC NEUROSCIENCES GMBH (DE) 2009-08-06 WO disclosed