SCHEMBL4180617

SCHEMBL4180617

CS(=O)(=O)c1ccc(-c2nnc(-c3ccc(C(F)(F)F)cc3C(N)c3ccncc3)[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.39
PTGS1 P23219 1/20 0.38
MAPK11 Q15759 2/20 0.37
MAPK14 Q16539 2/20 0.37
IDO1 P14902 2/20 0.37
TDO2 P48775 1/20 0.37
MAPK13 O15264 1/20 0.37
RAF1 P04049 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK12 P53778 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ALOX5 P09917 1/20 0.37
CSNK1A1 P48729 1/20 0.37
CSNK1D P48730 1/20 0.37
CSNK1E P49674 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CSNK1A1L Q8N752 1/20 0.37
SCD O00767 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
SLC22A12 Q96S37 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4177977 0.79 PTGS2 (0.43) PTGS2PTGS1IDO1TDO2PTGDR2
SCHEMBL4180618 0.76 PTGS2 (0.52) PTGS2PTGS1MAPK11MAPK14MAPK13
SCHEMBL4182513 0.74 GAA (0.42) PTGS2IDO1ALDH1A1SMN1; SMN2PTGDR2
SCHEMBL4177413 0.67 NPY5R (0.37) MAPK11MAPK14IDO1MAPK13RAF1
SCHEMBL4171248 0.66 HDAC8 (0.34) MAPK11MAPK14IDO1MAPK13RAF1
SCHEMBL4180993 0.65 PTGS2 (0.47) PTGS2PTGS1SCD
SCHEMBL7506839 0.65 PTGS2 (0.72) PTGS2PTGDR2
SCHEMBL15245162 0.64 SCD (0.55) SCD
SCHEMBL863126 0.64 PTGS2 (0.68) PTGS2
SCHEMBL4171111 0.63 TEK (0.44) MAPK11MAPK14MAPK13RAF1MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090318438-A1 Heterocyclic compounds and their use as anticancer agents CHEN XIAOLING 2009-12-24 US disclosed
US-20090048301-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS ANTICANCER AGENTS IMCLONE SYSTEMS INCORPORATED (US) 2009-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048301-A1 HETEROCYCLIC COMPOUNDS AND THEIR USE AS ANTICANCER AGENTS TP53, MCL1, VHL PTGS2 1129/4885PTGS1 835/4885MAPK11 1962/4885
US-20090318438-A1 Heterocyclic compounds and their use as anticancer agents TP53, MCL1, VHL PTGS2 1129/4885PTGS1 835/4885MAPK11 1962/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.