SCHEMBL4190738

SCHEMBL4190738

O=C(Nc1ccc(C=CCN2CCOCC2)cc1C1=CCCCC1)C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 14/20 0.48
KIT P10721 3/20 0.44
NTRK1 P04629 1/20 0.41
LCK P06239 1/20 0.41
CYP3A4 P08684 1/20 0.41
AXL P30530 1/20 0.41
FLT3 P36888 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4188266 0.83 CSF1R (0.43) CSF1RKIT
SCHEMBL4189779 0.81 CSF1R (0.67) CSF1RKITNTRK1LCKCYP3A4
SCHEMBL5650146 0.80 CSF1R (0.66) CSF1RKITCYP3A4
SCHEMBL2913376 0.79 CSF1R (0.64) CSF1RKITNTRK1LCKCYP3A4
SCHEMBL4185481 0.76 CSF1R (0.46) CSF1RKIT
SCHEMBL3083546 0.69 CSF1R (0.60) CSF1RKIT
SCHEMBL3086038 0.69 CSF1R (0.63) CSF1RKITNTRK1LCKCYP3A4
SCHEMBL5651779 0.69 CSF1R (0.63) CSF1RKIT
SCHEMBL3082962 0.69 CSF1R (0.57) CSF1R
SCHEMBL2913128 0.69 CSF1R (0.64) CSF1RKITNTRK1LCKCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2021329-A1 INHIBITORS OF C-FMS KINASE Janssen Pharmaceutica, N.V. (BE) 2009-02-11 EP disclosed
WO-2007124318-A1 INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2007-11-01 WO disclosed