SCHEMBL4190780

SCHEMBL4190780

O=C(NCC1CCCCC1)c1cc(Cl)ccc1NC(=O)c1cccc2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 8/20 1.00
CNR2 P34972 7/20 1.00
MEN1 O00255 1/20 0.56
RAB9A P51151 1/20 0.56
KMT2A Q03164 1/20 0.56
NPC1 O15118 2/20 0.56
ALDH1A1 P00352 2/20 0.56
BCHE P06276 1/20 0.50
CCR3 P51677 1/20 0.50
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
EPHX1 P07099 1/20 0.48
EPHX2 P34913 1/20 0.48
CHRM1 P11229 2/20 0.48
CHRM2 P08172 1/20 0.48
CHRM4 P08173 1/20 0.48
CHRM3 P20309 1/20 0.48
GFER P55789 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4194303 0.95 CNR1 (0.90) CNR1CNR2MEN1RAB9AKMT2A
SCHEMBL4191417 0.90 CNR1 (0.82) CNR1CNR2MEN1RAB9AKMT2A
SCHEMBL4198267 0.89 CNR2 (0.79) CNR1CNR2NPC1ALDH1A1CYP1A2
SCHEMBL5224040 0.88 CNR1 (0.78) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4190849 0.88 CNR1 (0.78) CNR1CNR2MEN1RAB9AKMT2A
SCHEMBL5314765 0.88 CNR1 (0.78) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL4198495 0.85 CNR1 (0.75) CNR1CNR2NPC1CCR3
SCHEMBL4193303 0.85 CNR1 (0.75) CNR1CNR2
SCHEMBL5220662 0.85 CNR1 (0.74) CNR1CNR2NPC1ALDH1A1BCHE
SCHEMBL5224036 0.85 CNR1 (0.74) CNR1CNR2NPC1ALDH1A1BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP claimed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO claimed
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP disclosed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO disclosed