SCHEMBL419195

SCHEMBL419195

Oc1ccc(-c2ccco2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 5/20 0.61
ERN1 O75460 2/20 0.50
ESR1 P03372 2/20 0.47
ESR2 Q92731 2/20 0.47
LPL P06858 1/20 0.47
LIPG Q9Y5X9 1/20 0.47
POLB P06746 3/20 0.46
KDM4E B2RXH2 2/20 0.46
MEN1 O00255 2/20 0.46
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 2/20 0.46
TSHR P16473 1/20 0.46
ADORA2A P29274 1/20 0.45
ADORA2B P29275 1/20 0.45
ADORA1 P30542 1/20 0.45
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
THRB P10828 1/20 0.44
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27639351 0.98 TAAR1 (0.59) TAAR1ERN1ESR1ESR2LPL
SCHEMBL14542115 0.88 TAAR1 (0.59) TAAR1ERN1ESR1ESR2LPL
SCHEMBL394300 0.87 TAAR1 (0.76) TAAR1ERN1LPLLIPGPOLB
SCHEMBL30487922 0.85 TAAR1 (0.73) TAAR1ERN1LPLLIPGPOLB
SCHEMBL244155 0.79
SCHEMBL6067949 0.79 ERN1 (0.49) TAAR1ERN1ESR1ESR2POLB
SCHEMBL3468357 0.79 TAAR1 (0.41) TAAR1ERN1ESR1ESR2LPL
SCHEMBL7404185 0.78 TAAR1 (0.64) TAAR1LPLLIPGPOLBKDM4E
SCHEMBL28323221 0.77 TAAR1 (0.62) TAAR1ERN1LPLLIPGPOLB
SCHEMBL162083 0.77 TAAR1 (0.62) TAAR1LPLLIPGPOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113582949-B Oxygen bridge bicyclo- [2.2.1] -heptene compound containing different covalent warhead structures and preparation and application thereof 武汉大学 2023-06-30 CN claimed
CN-113582949-A Oxygen-bridged bicyclo- [2.2.1] -heptene compound containing different covalent warhead structures and preparation and application thereof 武汉大学 2021-11-02 CN claimed
CN-108864127-B Oxidobicycloheptene sulfonamide compound with different alkyl chain lengths as well as preparation method and application thereof 武汉大学 2020-06-23 CN claimed
CN-107188896-B Oxocycloheptene compound containing resveratrol group and preparation and use method thereof 苏州楚凯药业有限公司 2020-04-03 CN claimed
CN-109942595-A Oxygen bridge containing different functionalities side-chain structure is bicyclic-[2.2.1]-heptan vinyl compound and its preparation and application 武汉大学 2019-06-28 CN claimed
CN-108864127-A A kind of oxygen bridge double-heptene sulfamide compound and the preparation method and application thereof containing different alkyl chain lengths 武汉大学 2018-11-23 CN claimed
CN-105111244-B Bicyclic [2.2.1] vinyl compound in heptan of ferrocene oxygen bridge 铱诺(武汉)药业有限公司 2018-02-09 CN claimed
CN-103596943-B Hydantoin derivatives useful as KV3 inhibitors 奥蒂福尼疗法有限公司 2016-10-12 CN claimed
CN-100522128-C Keratin dyeing compounds, keratin dyeing compositions containing them and their use PROCTER & GAMBLE (US) 2009-08-05 CN claimed
CN-115850294-B Oxygen bridge bicyclo- [2.2.1] -heptene compound containing selenocyano side chain, and preparation method and application thereof 武汉大学 2024-06-28 CN disclosed
CN-115557965-B PROTACs compound for dual targeting degradation of estrogen receptor alpha and aromatizing enzyme and application thereof 武汉大学 2024-03-19 CN disclosed
CN-113582949-B Oxygen bridge bicyclo- [2.2.1] -heptene compound containing different covalent warhead structures and preparation and application thereof 武汉大学 2023-06-30 CN disclosed
CN-114560867-B Oxygen bridge bicycloheptene sulfonate compound containing five-membered nitrogen heterocycle and application thereof in preparation of breast cancer resisting drugs 武汉大学 2023-06-06 CN disclosed
CN-113773283-B Oxidobicycloheptene sulfonamide compound containing hydrophobic label and application thereof 武汉大学 2023-04-07 CN disclosed
CN-1709241-A Intravenous injection stable concertrated clear solution containing rifamycin after dilution SUZHOU CHANGZHENG XINKAI PHARM (CN) 2005-12-21 CN disclosed
US-4857539-A Heterocyclic substituted-phenoxyalkylisoxazoles as antiviral useful agents STERLING DRUG INC. (US) 1989-08-15 US disclosed
EP-0207453-A2 Heterocyclic substituted-phenoxyalkyl-isoxazoles and-furans, their preparation and use as antiviral agents STERLING WINTHROP INC. (US) 1987-01-07 EP disclosed
US-4431831-A ANTIINFLAMMATORY AND ANTIARTHRITIC AGENTS RIKER LABORATORIES, INC. (US) 1984-02-14 US disclosed
EP-0080356-A2 Substituted furans RIKER LABORATORIES, INC. (US) 1983-06-01 EP disclosed
US-4357345-A ANTIINFLAMMATORY AGENTS RIKER LABORATORIES, INC. (US) 1982-11-02 US disclosed