SCHEMBL4194768

SCHEMBL4194768

Cc1cccc(-n2nc(CC(NC(=O)O)C(C)(C)C)cc2Sc2ccc(Cl)nc2)c1F

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2B Q13224 1/20 0.31
SLC16A3 O15427 1/20 0.31
SLC16A1 P53985 1/20 0.31
CTSA P10619 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3814311 0.94 RIPK1 (0.36) RXRAGRIN1GRIN2BSLC16A3SLC16A1
SCHEMBL3703229 0.94 SLC16A3 (0.32) SLC16A3SLC16A1CTSA
SCHEMBL3692814 0.91 SCN9A (0.35) RXRAGRIN1GRIN2BSLC16A3SLC16A1
SCHEMBL3700535 0.90 KCNQ3 (0.31) SLC16A3SLC16A1CTSA
SCHEMBL3709565 0.90 CTSA (0.36) SLC16A3SLC16A1CTSA
SCHEMBL3029599 0.88 SLC16A3 (0.37) SLC16A3SLC16A1
SCHEMBL3698043 0.88 KCNQ3 (0.32)
SCHEMBL3703720 0.86 KCNQ3 (0.31)
SCHEMBL3812496 0.86 KCNQ3 (0.33) RXRAGRIN1GRIN2B
SCHEMBL3695015 0.86 DHODH (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed