SCHEMBL4195546

SCHEMBL4195546

NC1=C2CCNCCC2NC=N1

nearest known ligand 0.31

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31
ALOX15 P16050 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2340625 0.64
Hydrochloric Acid SCHEMBL4401072 0.55
SCHEMBL128779 0.52
SCHEMBL2550391 0.52
SCHEMBL21998528 0.51
SCHEMBL31438848 0.50 HRH4 (0.42) HRH4MEN1ALDH1A1MAPTPKM
SCHEMBL719964 0.49 ADCY6 (0.56) MEN1ALDH1A1MAPTPKMKMT2A
SCHEMBL24067500 0.47 SLC18A3 (0.64) HRH4MAPT
SCHEMBL15221241 0.47
SCHEMBL21718408 0.47

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024368-A2 6,7,8,9-TETRAHYDRO-5H-PYRIMIDO[4,5-D]AZEPIN-4-YL]-AMINE DERIVATIVES AS MODULATORS OF TRPV1 FOR THE TREATMENT OF PAIN Janssen Pharmaceutica, N.V. (BE) 2009-02-18 EP claimed
WO-2007109355-A2 6,7,8, 9 -TETRAHYDRO- 5H- PYRIMIDO [4, 5-D] AZEPIN-4-YL] -AMINE DERIVATIVES AS MODULATORS OF TRPVL FOR THE TREATMENT OF PAIN JANSSEN PHARMACEUTICA N.V. (BE) 2007-09-27 WO claimed