SCHEMBL4195660

SCHEMBL4195660

Brc1ccc2[nH]c3c(c2c1)CCC[C@H]3NC1Cc2ccccc2C1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.67
KCNH2 Q12809 1/20 0.61
RB1 P06400 7/20 0.58
DHODH Q02127 2/20 0.57
CCNB2 O95067 1/20 0.48
CDK1 P06493 1/20 0.48
CCNB1 P14635 1/20 0.48
CCNB3 Q8WWL7 1/20 0.48
MAPT P10636 3/20 0.47
ALOX15 P16050 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
GLA P06280 1/20 0.47
KMT2A Q03164 1/20 0.47
CDC42 P60953 1/20 0.47
BRD3 Q15059 2/20 0.43
GAA P10253 1/20 0.43
CASP6 P55212 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4196044 1.00 CYP2D6 (0.67) CYP2D6KCNH2RB1DHODHCCNB2
SCHEMBL4163592 1.00 CYP2D6 (0.67) CYP2D6KCNH2RB1DHODHCCNB2
Hydrochloric Acid SCHEMBL4165683 0.99 CYP2D6 (0.65) CYP2D6KCNH2RB1DHODHCCNB2
Hydrochloric Acid SCHEMBL4148242 0.99 CYP2D6 (0.65) CYP2D6KCNH2RB1DHODHCCNB2
SCHEMBL4194091 0.91 RB1 (0.58) CYP2D6KCNH2RB1DHODHCCNB2
Hydrochloric Acid SCHEMBL4157051 0.90 RB1 (0.59) CYP2D6KCNH2RB1DHODHCCNB2
SCHEMBL21998619 0.87 RB1 (0.68) CYP2D6KCNH2RB1DHODHMAPT
SCHEMBL4187335 0.86 GAA (0.59) CYP2D6KCNH2RB1MAPTALOX15
SCHEMBL5394699 0.86 RB1 (0.69) CYP2D6KCNH2RB1DHODHMAPT
SCHEMBL4188706 0.86 RB1 (0.78) CYP2D6KCNH2RB1MAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1658068-B1 NOVEL CYCLOALKYL[B] CONDENSED INDOLES SMITHKLINE BEECHAM CORP (US) 2009-02-18 EP claimed
US-7622494-B2 Chemical compounds SMITHKLINE BEECHAM CORPORATION (US) 2009-11-24 US disclosed
US-7622494-B2 Chemical compounds SMITHKLINE BEECHAM CORPORATION (US) 2009-11-24 US disclosed
US-20090170923-A1 HCV INHIBITORS SMITHKLINE BEECHAM CORPORATION 2009-07-02 US disclosed
US-20090170923-A1 HCV INHIBITORS SMITHKLINE BEECHAM CORPORATION 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170923-A1 HCV INHIBITORS HAVCR2, MAVS, EIF2AK2 CYP2D6 994/4885KCNH2 4356/4885RB1 4460/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.