SCHEMBL4195752

SCHEMBL4195752

CCN(C1CCc2cc(C(=O)Nc3ccccc3NC(=O)O)ccc21)S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.46
MAPT P10636 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 2/20 0.42
POLB P06746 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.40
CYP3A4 P08684 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4186907 0.91 CA12 (0.50) APEX1MAPTSMN1; SMN2MEN1LMNA
SCHEMBL13653115 0.89 APEX1 (0.41) APEX1MAPTSMN1; SMN2MEN1LMNA
SCHEMBL4174953 0.87 CA12 (0.50) APEX1MAPTTP53CA12CA9
SCHEMBL4195612 0.86 CA12 (0.45) APEX1MAPTSMN1; SMN2MEN1LMNA
SCHEMBL4187089 0.84 CA12 (0.49) LMNACA12CA9ALDH1A1KDM4E
SCHEMBL4195619 0.83 CA12 (0.44) APEX1SMN1; SMN2MEN1LMNATSHR
SCHEMBL4185822 0.83 HDAC1 (0.50) MAPTCA12CA9
SCHEMBL4189530 0.82 KMT2A (0.41) APEX1MAPTMEN1LMNAKMT2A
SCHEMBL4197907 0.82 HDAC1 (0.45) MAPTSMN1; SMN2MEN1KMT2ACA12
SCHEMBL4185649 0.81 CA12 (0.43) MAPTSMN1; SMN2MEN1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090247590-A1 Indane amides BAYER PHARMACEUTICLAS CORPORATION (US) 2009-10-01 US disclosed
EP-1802577-A1 INDANE AMIDES WITH ANTIPROLIFERATIVE ACTIVITY Bayer Pharmaceuticals Corporation (US) 2007-07-04 EP disclosed
WO-2006062580-A1 INDANE AMIDES WITH ANTIPROLIFERATIVE ACTIVITY BAYER PHARMACEUTICALS CORPORATION (US) 2006-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090247590-A1 Indane amides MKI67, PPIP5K2, CCNA1 APEX1 732/4885MAPT 1308/4885SMN1; SMN2 3677/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.