SCHEMBL4196232

SCHEMBL4196232

Nc1ncc(-c2cc(Cl)ccc2Cl)c(N)n1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 7/20 0.61
HTR2B P41595 1/20 0.54
PDE4D Q08499 1/20 0.54
FGFR1 P11362 1/20 0.48
SRC P12931 1/20 0.48
SCN10A Q9Y5Y9 1/20 0.47
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
ADORA1 P30542 2/20 0.44
ADORA2A P29274 1/20 0.44
AGPAT2 O15120 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388588 0.86 DHFR (0.59) DHFRFGFR1SRCMAPTADORA1
SCHEMBL168973 0.79 SCN2A (0.57) DHFRFGFR1SRCSCN10AADORA1
SCHEMBL30413525 0.79 SCN2A (0.57) DHFRFGFR1SRCSCN10AADORA1
SCHEMBL4186547 0.79 DHFR (0.56) DHFRFGFR1SRCSCN10AADORA1
SCHEMBL1388506 0.77 DHFR (0.67) DHFRMEN1HTTKMT2A
SCHEMBL29913206 0.77 DHFR (0.67) DHFRMEN1HTTKMT2A
SCHEMBL1388267 0.76 DHFR (1.00) DHFRFGFR1SRCADORA1ADORA2A
SCHEMBL263262 0.75 SCN10A (0.56) HTR2BPDE4DSCN10AMEN1MAPT
SCHEMBL1388562 0.75 DHFR (1.00) DHFRFGFR1SRCADORA1ADORA2A
SCHEMBL29913330 0.75 DHFR (1.00) DHFRFGFR1SRCADORA1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2032543-A1 2-ANILINO-4-AMINOALKYLENEAMINOPYRIMIDINES Boehringer Ingelheim International GmbH (DE) 2009-03-11 EP disclosed
WO-2007146977-A1 2-ANILINO-4-AMINOALKYLENEAMINOPYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-12-21 WO disclosed