SCHEMBL4196590

SCHEMBL4196590

O=C(Nc1ccc(Cl)cc1C(=O)NCC1CCCCC1)c1cnc2ccccc2n1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.66
CNR1 P21554 6/20 0.66
NPC1 O15118 1/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4195914 0.87 CNR1 (0.69) CNR2CNR1NPC1CYP2C9CYP1A2
SCHEMBL4204619 0.87 CNR2 (0.66) CNR2CNR1NPC1CYP3A4CYP2C9
SCHEMBL27684178 0.81 CNR1 (0.72) CNR2CNR1NPC1POLBTSHR
SCHEMBL4190614 0.81 CNR2 (0.61) CNR2CNR1NPC1CYP3A4CYP2C9
SCHEMBL4193009 0.81 CNR2 (0.69) CNR2CNR1NPC1CYP3A4CYP2C9
SCHEMBL4198495 0.79 CNR1 (0.75) CNR2CNR1NPC1POLBTSHR
SCHEMBL4193303 0.79 CNR1 (0.75) CNR2CNR1
SCHEMBL4188684 0.79 CNR1 (0.72) CNR2CNR1NPC1POLBTSHR
SCHEMBL4188696 0.79 CNR2 (0.63) CNR2CNR1NPC1POLBTSHR
SCHEMBL4190780 0.79 CNR1 (1.00) CNR2CNR1NPC1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP claimed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO claimed
EP-1756044-A1 THERAPEUTIC COMPOUNDS AstraZeneca AB (SE) 2007-02-28 EP disclosed
WO-2005115972-A1 THERAPEUTIC COMPOUNDS ASTRAZENECA AB (SE) 2005-12-08 WO disclosed