SCHEMBL4200618

SCHEMBL4200618

CCC(CC)n1ccc2cnc(Nc3ccc(N4CCC(CC=O)CC4)cc3)nc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 17/20 0.50
CCND1 P24385 10/20 0.50
CCND2 P30279 9/20 0.50
CCND3 P30281 9/20 0.50
AURKA O14965 7/20 0.47
CDK1 P06493 3/20 0.47
INSR P06213 1/20 0.47
PDGFRB P09619 1/20 0.47
SRC P12931 1/20 0.47
PDGFRA P16234 1/20 0.47
FLT1 P17948 1/20 0.47
FLT4 P35916 1/20 0.47
KDR P35968 1/20 0.47
CDK7 P50613 1/20 0.47
NTRK2 Q16620 1/20 0.47
FGFR4 P22455 5/20 0.47
CDK2 P24941 5/20 0.46
CCNE2 O96020 4/20 0.46
CCNE1 P24864 4/20 0.46
CCNA2 P20248 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4200615 0.84 CDK4 (0.49) CDK4CCND1CCND2CCND3AURKA
SCHEMBL7713198 0.83 CDK4 (0.62) CDK4CCND1CCND2CCND3AURKA
SCHEMBL4195694 0.83 CDK4 (0.50) CDK4CCND1CCND2CCND3AURKA
SCHEMBL4200620 0.82 CDK4 (0.51) CDK4CCND1CCND2CCND3AURKA
SCHEMBL4342366 0.82 CDK4 (0.60) CDK4CCND1CCND2CCND3CDK1
SCHEMBL7706847 0.80 ALK (0.58) CDK4CCND1CDK2CCNE1
SCHEMBL11977054 0.80 SYK (0.55) CDK4CCND1CCND2CCND3AURKA
SCHEMBL4515832 0.76 CCND3 (0.57) CDK4CCND1CCND2CCND3CDK2
SCHEMBL11976956 0.73 JAK2 (0.57)
SCHEMBL11977047 0.73 CDK4 (0.62) CDK4CCND1CCND2CCND3CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029145-A2 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES Novartis Ag (CH) 2009-03-04 EP disclosed
WO-2007140222-A2 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2007-12-06 WO disclosed