SCHEMBL4207983

SCHEMBL4207983

O=c1[nH]cnc2c1sc1cc(Br)ccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 6/20 0.49
PIM3 Q86V86 5/20 0.49
CHEK1 O14757 1/20 0.49
AKT1 P31749 1/20 0.49
FLT3 P36888 1/20 0.49
PIM2 Q9P1W9 3/20 0.48
CDC7 O00311 2/20 0.48
CSNK2A1 P68400 2/20 0.48
POLB P06746 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
CSNK2A2 P19784 1/20 0.48
CSNK2B P67870 1/20 0.48
CSNK2A3 Q8NEV1 1/20 0.48
CLK4 Q9HAZ1 3/20 0.44
DAPK3 O43293 2/20 0.44
PRKD3 O94806 2/20 0.44
GSK3A P49840 2/20 0.44
GSK3B P49841 2/20 0.44
DYRK1A Q13627 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4219756 0.88 PIM1 (0.53) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL4215069 0.82 ALDH1A1 (0.53) PIM1PIM3PIM2CDC7CSNK2A1
SCHEMBL4207625 0.82 PARP1 (0.49) PIM1PIM3PIM2CDC7CSNK2A1
SCHEMBL4208127 0.79 LIMK1 (0.59) PIM1PIM3PIM2CDC7CSNK2A1
SCHEMBL4208864 0.78 KRAS (0.51) PIM1PIM3PIM2CDC7CSNK2A1
SCHEMBL2307979 0.77 HTT (0.51) PIM1PIM3CHEK1AKT1FLT3
SCHEMBL4208101 0.75 PARP1 (0.41) PIM1PIM3PIM2CDC7CSNK2A1
SCHEMBL2302798 0.75 KDM4A (0.51) PIM1PIM3PIM2CDC7CSNK2A1
SCHEMBL4207979 0.73 PARP1 (0.53) PIM1PIM3CHEK1PIM2CDC7
SCHEMBL4213078 0.73 PIM1 (0.59) PIM1PIM3PIM2CDC7CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090030196-A1 PIM KINASE INHIBITORS AS CANCER CHEMOTHERAPEUTICS ABBOTT LABORATORIES (US) 2009-01-29 US claimed
US-20090030196-A1 PIM KINASE INHIBITORS AS CANCER CHEMOTHERAPEUTICS ABBOTT LABORATORIES (US) 2009-01-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090030196-A1 PIM KINASE INHIBITORS AS CANCER CHEMOTHERAPEUTICS PIM1, PIM3, PIM2 PIM1 1/4885PIM3 2/4885CHEK1 38/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.