Cyclopropane

Cyclopropane

SCHEMBL4211055

C1CC1.O=C(O)Nc1cccc2c1C(=O)N(C(CC(=O)NO)c1ccc(OC(F)F)c(OC(F)F)c1)C2

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPT P10636 7/20 0.41
TDP1 Q9NUW8 1/20 0.40
TP53 P04637 5/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclopropane SCHEMBL4206831 0.94 TP53 (0.46) MEN1KMT2AMAPTTDP1TP53
Cyclopropane SCHEMBL4206835 0.91 PDE4A (0.41) MEN1KMT2AMAPTTDP1TP53
Cyclopropane SCHEMBL4204875 0.89 MEN1 (0.39) MEN1KMT2AMAPTTDP1TP53
SCHEMBL1144306 0.89 MAPT (0.40) MEN1KMT2AMAPTTDP1TP53
SCHEMBL1143447 0.85 PDE4A (0.49) MEN1KMT2AMAPTTP53
Cyclopropane SCHEMBL4200950 0.85 PDE4B (0.51) MEN1KMT2ATP53
Cyclopropane SCHEMBL15252535 0.85 TP53 (0.52) MEN1KMT2AMAPTTP53
SCHEMBL1143737 0.83 TP53 (0.44) MEN1KMT2AMAPTTP53
SCHEMBL1143956 0.82 MEN1 (0.39) MEN1KMT2AMAPTTP53
Cyclopropane SCHEMBL4206531 0.81 PDE4B (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1587474-B1 FLUOROALKOXY-SUBSTITUTED 1, 3-DIHYDRO-ISOINDOLYL COMPOUNDS AND THEIR PHARMACEUTICAL USES CELGENE CORP (US) 2009-11-18 EP claimed