SCHEMBL4211927

SCHEMBL4211927

CCOc1cccc(Cl)c1-c1cc(Cl)nc(N)n1

nearest known ligand 0.73

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 12/20 0.73
HSP90AB1 P08238 10/20 0.73
AGPAT2 O15120 2/20 0.45
KDM4E B2RXH2 1/20 0.44
ADCY10 Q96PN6 3/20 0.43
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3949271 0.85 HSP90AA1 (0.67) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL3940837 0.85 HSP90AA1 (1.00) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL3945723 0.84 HSP90AA1 (0.65) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL4225202 0.83 HSP90AA1 (0.64) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL3941512 0.81 DHFR (0.55) HSP90AA1HSP90AB1AGPAT2KDM4EADCY10
SCHEMBL3951313 0.77 HSP90AA1 (1.00) HSP90AA1HSP90AB1KDM4EADCY10NPC1
SCHEMBL4033797 0.76 HSP90AA1 (0.55) HSP90AA1HSP90AB1KDM4EMAPK1
SCHEMBL3941695 0.76 HSP90AA1 (0.55) HSP90AA1HSP90AB1
SCHEMBL4530414 0.76 HSP90AA1 (0.55) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL22501986 0.76 HSP90AA1 (0.66) HSP90AA1HSP90AB1KDM4EADCY10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090215777-A1 Pyrimidine Derivatives As HSP90 Inhibitors ASTEX THERAPEUTICS LTD. (GB) 2009-08-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090215777-A1 Pyrimidine Derivatives As HSP90 Inhibitors HSP90AB1, HSP90AB2P, HSP90B1 HSP90AA1 4/4885HSP90AB1 1/4885AGPAT2 4537/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.