SCHEMBL4214955

SCHEMBL4214955

Cc1cccnc1CNC(CCCN)Cc1ncccc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 5/20 0.41
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
ADORA2A P29274 9/20 0.34
ADORA1 P30542 8/20 0.34
CHRM2 P08172 2/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
CYP1A2 P05177 2/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
ABCB11 O95342 1/20 0.33
ESR1 P03372 1/20 0.33
PGR P06401 1/20 0.33
ADRB2 P07550 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2082171 0.92 ADORA2A (0.41) CXCR4MAOAMAOBHSP90AA1HSP90AB1
SCHEMBL2083908 0.91 ADORA2A (0.38) CXCR4MAOAMAOBHSP90AA1HSP90AB1
SCHEMBL2085159 0.91 CXCR4 (0.38) CXCR4MAOAMAOBHSP90AA1HSP90AB1
SCHEMBL2083555 0.89 CXCR4 (0.39) CXCR4MAOAMAOBHSP90AA1HSP90AB1
SCHEMBL2084233 0.88 CXCR4 (0.42) CXCR4MAOAMAOBHSP90AA1HSP90AB1
SCHEMBL2084154 0.87 ADORA2A (0.37) CXCR4ADORA2AADORA1ADRB2
SCHEMBL2085140 0.87 AGBL2 (0.36) CXCR4MAOAMAOBADORA2AADORA1
SCHEMBL2084251 0.85 HRH1 (0.39) CXCR4MAOAMAOBHSP90AA1HSP90AB1
SCHEMBL2085079 0.85 CXCR4 (0.35) CXCR4MAOAMAOBADORA2AADORA1
SCHEMBL2081740 0.85 CXCR4 (0.35) CXCR4MAOAMAOBADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed