SCHEMBL4215022

SCHEMBL4215022

CCCOc1ccc(-c2nn(C)c3nc(N)ncc23)cc1F

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 10/20 0.74
TLR9 Q9NR96 10/20 0.69
TLR8 Q9NR97 10/20 0.69
BTK Q06187 4/20 0.42
PIK3CA P42336 2/20 0.39
MTOR P42345 2/20 0.39
RICTOR Q6R327 1/20 0.39
RPTOR Q8N122 1/20 0.39
MAPKAP1 Q9BPZ7 1/20 0.39
MLST8 Q9BVC4 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PDE5A O76074 1/20 0.37
PIK3CD O00329 1/20 0.37
ABL1 P00519 1/20 0.37
EGFR P00533 1/20 0.37
HCK P08631 1/20 0.37
SRC P12931 1/20 0.37
KDR P35968 1/20 0.37
PIK3CB P42338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4214625 0.91 TLR7 (0.74) TLR7TLR9TLR8BTKPIK3CA
SCHEMBL4228277 0.91 TLR7 (0.70) TLR7TLR9TLR8PIK3CAMTOR
SCHEMBL4044815 0.90 TLR7 (0.72) TLR7TLR9TLR8PIK3CAMTOR
SCHEMBL4275196 0.89 TLR7 (0.74) TLR7TLR9TLR8BTKPIK3CA
SCHEMBL4226497 0.87 TLR7 (0.79) TLR7TLR9TLR8BTK
SCHEMBL4047282 0.86 TLR7 (0.67) TLR7TLR9TLR8PIK3CAMTOR
SCHEMBL4046635 0.86 TLR7 (0.67) TLR7TLR9TLR8PIK3CAMTOR
SCHEMBL4221225 0.85 TLR7 (1.00) TLR7TLR9TLR8KDR
SCHEMBL4223404 0.84 TLR7 (0.75) TLR7TLR9TLR8KDM4E
SCHEMBL4219300 0.84 TLR7 (0.65) TLR7TLR9TLR8KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2026811-A1 PYRAZOLO [3, 4-D]PYRIMIDINE DERIVATIVES USEFUL TO TREAT RESPIRATORY DISORDERS Novartis AG (CH) 2009-02-25 EP disclosed
WO-2007134828-A1 PYRAZOLO [3, 4-D] PYRIMIDINE DERIVATIVES USEFUL TO TREAT RESPIRATORY DISORDERS NOVARTIS AG (CH) 2007-11-29 WO disclosed