SCHEMBL4221297

SCHEMBL4221297

COc1nc2ccn(C)c2cc1C1=CCN(C(=O)O)CC1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
QDPR P09417 2/20 0.36
SUV39H2 Q9H5I1 5/20 0.35
TDP1 Q9NUW8 1/20 0.34
PDE10A Q9Y233 3/20 0.33
CCNT1 O60563 1/20 0.33
CDK9 P50750 1/20 0.33
MAPT P10636 1/20 0.32
JAK1 P23458 1/20 0.32
PARP1 P09874 1/20 0.32
SCD O00767 1/20 0.32
SCD5 Q86SK9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5101441 0.87 PDK4 (0.48) PDE10AJAK1
SCHEMBL22119718 0.75 QDPR (0.38) QDPRSUV39H2TDP1PDE10ACCNT1
SCHEMBL16875073 0.73 BTK (0.41)
SCHEMBL16875075 0.73 BTK (0.41)
SCHEMBL4219836 0.73 PDK4 (0.46) PDE10AJAK1
SCHEMBL16992066 0.71 PDE10A (0.46) PDE10ACCNT1CDK9
SCHEMBL6812301 0.70 SLC6A4 (0.44)
SCHEMBL4335947 0.69 QDPR (0.48) QDPRCCNT1CDK9MAPT
SCHEMBL22119654 0.68 QDPR (0.38) QDPRSUV39H2TDP1MAPT
SCHEMBL16422788 0.68 SUV39H2 (0.40) QDPRSUV39H2TDP1MAPTSCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013214-A2 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS Bristol-Myers Squibb Company (US) 2009-01-14 EP disclosed
WO-2007131020-A2 CONSTRAINED COMPOUNDS AS CGRP-RECEPTOR ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-15 WO disclosed