Known targets — ChEMBL curated mechanism
SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9A
The experimentally established mechanism targets of Mexiletine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.
Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | SCN5A known ✓ | Q14524 | 3/20 | 1.00 |
| ▸ | SCN1A known ✓ | P35498 | 2/20 | 1.00 |
| ▸ | SCN9A known ✓ | Q15858 | 2/20 | 1.00 |
| ▸ | SCN4A known ✓ | P35499 | 10/20 | 0.96 |
| ▸ | SCN7A known ✓ | Q01118 | 1/20 | 0.96 |
| ▸ | SCN2A known ✓ | Q99250 | 1/20 | 0.96 |
| ▸ | SCN3A known ✓ | Q9NY46 | 1/20 | 0.96 |
| ▸ | SCN11A known ✓ | Q9UI33 | 1/20 | 0.96 |
| ▸ | SCN8A known ✓ | Q9UQD0 | 1/20 | 0.96 |
| ▸ | SCN10A known ✓ | Q9Y5Y9 | 1/20 | 0.96 |
| ▸ | LMNA | P02545 | 3/20 | 1.00 |
| ▸ | CYP2D6 | P10635 | 3/20 | 0.96 |
| ▸ | CYP1A2 | P05177 | 2/20 | 0.96 |
| ▸ | CYP3A4 | P08684 | 2/20 | 0.96 |
| ▸ | NFKB1 | P19838 | 2/20 | 0.96 |
| ▸ | TSHR | P16473 | 2/20 | 0.96 |
| ▸ | MAOA | P21397 | 2/20 | 0.96 |
| ▸ | CYP2C9 | P11712 | 1/20 | 0.96 |
| ▸ | KCNK3 | O14649 | 1/20 | 0.96 |
| ▸ | CACNA1F | O60840 | 1/20 | 0.96 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Mexiletine SCHEMBL6521444 | 1.00 | SCN5A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| (S)-Mexiletine SCHEMBL3645798 | 1.00 | SCN5A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| Mexiletine SCHEMBL6665250 | 1.00 | SCN5A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| (R)-Mexiletine SCHEMBL29366590 | 1.00 | SCN5A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| (S)-Mexiletine SCHEMBL13046569 | 0.98 | SCN4A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| (R)-Mexiletine SCHEMBL16082 | 0.98 | SCN4A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| Mexiletine SCHEMBL8858385 | 0.98 | SCN4A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| Mexiletine SCHEMBL16081 | 0.98 | SCN4A (1.00) | SCN5ALMNASCN1ASCN9ASCN4A | |
| Mexiletine SCHEMBL1652207 | 0.94 | SCN4A (0.92) | SCN5ALMNASCN1ASCN9ASCN4A | |
| Mexiletine SCHEMBL8819167 | 0.88 | SCN4A (0.80) | SCN5ALMNASCN1ASCN9ASCN4A |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Appears in 4190 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-121585847-A | Screen projection processing method, device and storage medium | 长城汽车股份有限公司 | 2026-02-27 | — | — | CN | claimed |
| EP-4680201-A1 | COMPOSITIONS AND USES THEREOF FOR STABILIZATION OF BLOOD SAMPLE COMPONENTS | Streck LLC (US) | 2026-01-21 | — | — | EP | claimed |
| CN-119379366-B | Insurance advertisement dynamic loading method based on Internet | 星火智云(上海)科技发展有限公司 | 2025-06-13 | — | — | CN | claimed |
| CN-120020942-A | Audio generation method, system, device and storage medium | 北京字跳网络技术有限公司 | 2025-05-20 | — | — | CN | claimed |
| CN-119967204-A | Video and audio digital copyright encryption method, decryption method, system and device | 央视国际网络有限公司 | 2025-05-09 | — | — | CN | claimed |
| US-20250120930-A1 | COMPOSITIONS CONTAINING DOFETILIDE AND MEXILETINE AND USES THEREOF | FB-HRS, LLC | 2025-04-17 | — | — | US | claimed |
| CN-119759586-A | Resource allocation method based on event response | 众合云科信息技术集团有限公司 | 2025-04-04 | — | — | CN | claimed |
| CN-119728658-A | Audio broadcasting method, device, system, electronic equipment and storage medium | 科大讯飞股份有限公司 | 2025-03-28 | — | — | CN | claimed |
| CN-119417661-A | Multimedia interaction method and system | 山东悦正达信用服务有限公司 | 2025-02-11 | — | — | CN | claimed |
| WO-2024192232-A9 | COMPOSITIONS AND USES THEREOF FOR STABILIZATION OF BLOOD SAMPLE COMPONENTS | STRECK LLC (US) | 2025-02-06 | — | — | WO | claimed |
| WO-1992013935-A1 | PHOSPHATE-FREE CLEANING AGENT | HENKEL KOMMANDITGESELLSCHAFT AUF AKTIEN (DE) | 1992-08-20 | — | — | WO | claimed |
| EP-0425428-A2 | Method for preparation of sodium silicates | HOECHST AKTIENGESELLSCHAFT (DE) | 1991-05-02 | — | — | EP | claimed |
| EP-0387251-A1 | USE OF FILLERS COATED WITH TRIALKOXYSILANES | NAINTSCH MINERALWERKE GESELLSCHAFT M.B.H. (AT) | 1990-09-19 | — | — | EP | claimed |
| EP-0293640-A2 | Process for the production of crystalline sodium silicates having a layer structure | HOECHST AKTIENGESELLSCHAFT (DE) | 1988-12-07 | — | — | EP | claimed |
| EP-0126795-B1 | METHOD FOR MANUFACTURING WELDED PIPES | KAWASAKI JUKOGYO KABUSHIKI KAISHA (JP) | 1988-06-01 | — | — | EP | claimed |
| EP-0082254-B1 | IMAGE FORMING APPARATUS | KABUSHIKI KAISHA TOSHIBA (JP) | 1986-03-12 | — | — | EP | claimed |
| EP-0034183-B1 | TYING UP MACHINE | Maschinenfabrik Gerd Mosca GmbH (DE) | 1983-05-11 | — | — | EP | claimed |
| EP-0054241-A1 | Connection of a mast foot to a sail-board | Marker, Hannes (DE) | 1982-06-23 | — | — | EP | claimed |
| EP-0034183-A1 | TYING UP MACHINE. | MOSCA G MASCHF (DE) | 1981-08-26 | — | — | EP | claimed |
| WO-1981000548-A1 | TYING UP MACHINE | MOSCA G MASCHF (DE) | 1981-03-05 | — | — | WO | claimed |