SCHEMBL4222930

SCHEMBL4222930

CC(=O)N1CCC[C@H]1C(=O)N1CC(=O)[C@@H]2C1CCN2C(=O)[C@H](CC(C)C)NC(=O)c1ccc(N(C)C)cc1

nearest known ligand 0.71

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.71
CTSS P25774 1/20 0.42
ACE P12821 2/20 0.38
STAT3 P40763 4/20 0.38
CAPN1 P07384 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSB P07858 1/20 0.37
CCR1 P32246 1/20 0.36
ACE2 Q9BYF1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5941389 1.00 CTSK (0.71) CTSKCTSSACESTAT3CAPN1
SCHEMBL4044347 1.00 CTSK (0.71) CTSKCTSSACESTAT3CAPN1
SCHEMBL4217216 1.00 CTSK (0.71) CTSKCTSSACESTAT3CAPN1
SCHEMBL4042741 0.98 CTSK (0.70) CTSKCTSSACESTAT3CAPN1
SCHEMBL4045507 0.92 CTSK (0.60) CTSKCTSSACESTAT3CAPN1
SCHEMBL4364104 0.91 CTSK (0.82) CTSKCTSSKMT2ACTSBCCR1
SCHEMBL4364108 0.91 CTSK (0.82) CTSKCTSSKMT2ACTSBCCR1
SCHEMBL4364101 0.91 CTSK (0.82) CTSKCTSSKMT2ACTSBCCR1
SCHEMBL5941936 0.91 CTSK (0.82) CTSKCTSSKMT2ACTSBCCR1
SCHEMBL4042535 0.90 CTSK (0.58) CTSKCTSSACESTAT3CAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2051974-A1 TETRAHYDROBENZOTHIOPHENE DERIVATIVES 4SC AG (DE) 2009-04-29 EP disclosed
WO-2008020045-A1 TETRAHYDROBENZOTHIOPHENE DERIVATIVES 4SC AG (DE) 2008-02-21 WO disclosed