SCHEMBL4223446

SCHEMBL4223446

CC(C)C[C@H](NC(=O)c1ccc(N(C)C)cc1)C(=O)N1CCC2[C@H]1C(=O)CN2C(=O)[C@@H](N)CC(C)(C)C

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.71
CTSS P25774 3/20 0.45
DPP4 P27487 1/20 0.38
CCR1 P32246 1/20 0.36
POLB P06746 1/20 0.35
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
CTSV O60911 2/20 0.34
CTSL P07711 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039017 1.00 CTSK (0.71) CTSKCTSSDPP4CCR1POLB
SCHEMBL5942287 1.00 CTSK (0.71) CTSKCTSSDPP4CCR1POLB
SCHEMBL4223449 1.00 CTSK (0.71) CTSKCTSSDPP4CCR1POLB
SCHEMBL5941439 0.93 CTSK (0.77) CTSKCTSSDPP4CCR1POLB
SCHEMBL4207543 0.93 CTSK (0.77) CTSKCTSSDPP4CCR1POLB
SCHEMBL4207538 0.93 CTSK (0.77) CTSKCTSSDPP4CCR1POLB
SCHEMBL5941962 0.93 CTSK (0.77) CTSKCTSSDPP4CCR1POLB
SCHEMBL4040277 0.93 CTSK (0.77) CTSKCTSSDPP4CCR1POLB
SCHEMBL5941958 0.93 CTSK (0.77) CTSKCTSSDPP4CCR1POLB
SCHEMBL4042133 0.92 CTSK (0.60) CTSKCTSSDPP4CCR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed