SCHEMBL4228997

SCHEMBL4228997

CC(C)(C)OC(=O)/C=C/c1c[nH]c(C(=O)O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
HSP90AA1 P07900 1/20 0.38
PKM P14618 1/20 0.38
ESR1 P03372 1/20 0.38
NR1H4 Q96RI1 4/20 0.36
TDP1 Q9NUW8 2/20 0.35
GABBR2 O75899 1/20 0.35
GABBR1 Q9UBS5 1/20 0.35
DAO P14920 1/20 0.34
CYP3A4 P08684 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
NR1I2 O75469 1/20 0.34
PGR P06401 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
CYP2C9 P11712 1/20 0.34
SLC6A2 P23975 1/20 0.34
TBXAS1 P24557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4228999 1.00 SMN1; SMN2 (0.38) SMN1; SMN2RAB9ANPC1HSP90AA1PKM
SCHEMBL1081773 0.87 ALDH1A1 (0.42) ESR1NR1H4CYP3A4LMNAHTT
SCHEMBL1006832 0.87 ALDH1A1 (0.42) ESR1NR1H4CYP3A4LMNAHTT
SCHEMBL1006833 0.87 ALDH1A1 (0.42) ESR1NR1H4CYP3A4LMNAHTT
SCHEMBL13845311 0.78 ESR1 (0.45) ESR1NR1H4GABBR2GABBR1CYP3A4
SCHEMBL4054983 0.78 ESR1 (0.45) ESR1NR1H4GABBR2GABBR1CYP3A4
SCHEMBL4054986 0.78 ESR1 (0.45) ESR1NR1H4GABBR2GABBR1CYP3A4
SCHEMBL13658710 0.77 TDP1 (0.50) SMN1; SMN2RAB9ANPC1HSP90AA1PKM
SCHEMBL4055672 0.75 CA12 (0.53) RAB9ANPC1ESR1NR1H4LMNA
SCHEMBL13845314 0.75 CA12 (0.53) RAB9ANPC1ESR1NR1H4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074092-A2 INHIBITORS OF D-AMINO ACID OXIDASE Sepracor Inc. (US) 2009-07-01 EP disclosed
WO-2008089453-A2 INHIBITORS OF D-AMINO ACID OXIDASE SEPRACOR INC. (US) 2008-07-24 WO disclosed