SCHEMBL4229534

SCHEMBL4229534

CCN(CC)CCCC(NC(=O)Nc1ccc(F)c(C)c1)c1ccc(C(=O)Nc2ccccc2N)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 12/20 0.46
HDAC1 Q13547 12/20 0.46
HDAC8 Q9BY41 3/20 0.46
HDAC2 Q92769 9/20 0.43
NCOR2 Q9Y618 6/20 0.43
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 1/20 0.42
TMEM97 Q5BJF2 6/20 0.41
SIGMAR1 Q99720 6/20 0.41
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
HTR1A P08908 1/20 0.39
CHRM5 P08912 1/20 0.39
ADRA2A P08913 1/20 0.39
CHRM1 P11229 1/20 0.39
ADRA2B P18089 1/20 0.39
CHRM3 P20309 1/20 0.39
DRD1 P21728 1/20 0.39
DRD5 P21918 1/20 0.39
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2383746 0.94 HDAC1 (0.47) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL2385454 0.92 UTS2R (0.45) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL4224033 0.91 HDAC1 (0.51) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL4223952 0.90 HDAC1 (0.46) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL4219358 0.90 HDAC3 (0.46) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL2385536 0.89 HDAC3 (0.43) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL4228901 0.89 HDAC1 (0.47) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL3234270 0.88 TMEM97 (0.38) HDAC3HDAC1HDAC2NCOR2TMEM97
SCHEMBL4229378 0.87 HDAC1 (0.48) HDAC3HDAC1HDAC8HDAC2NCOR2
SCHEMBL2386741 0.86 HDAC3 (0.43) HDAC3HDAC1HDAC8HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2133339-A1 NOVEL (2-AMINOPHENYL)PYRIDINECARBOXAMIDE DERIVATIVE HAVING UREA STRUCTURE Santen Pharmaceutical Co., Ltd (JP) 2009-12-16 EP disclosed