Cliprofen

Cliprofen

SCHEMBL42298

CC(C(=O)O)c1ccc(C(=O)c2cccs2)c(Cl)c1

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.63
HPGD P15428 4/20 0.63
ALDH1A1 P00352 4/20 0.63
CYP2C9 P11712 3/20 0.63
LMNA P02545 3/20 0.63
PTGS2 P35354 3/20 0.63
KDM4E B2RXH2 2/20 0.63
RXFP1 Q9HBX9 1/20 0.63
CHRM1 P11229 1/20 0.47
ALOX15 P16050 2/20 0.46
SMN1; SMN2 Q16637 4/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MAPT P10636 3/20 0.43
HSD17B10 Q99714 2/20 0.43
PSMD14 O00487 1/20 0.43
MMP2 P08253 1/20 0.43
HPGDS O60760 1/20 0.42
AKR1C3 P42330 3/20 0.41
AKR1C2 P52895 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cliprofen SCHEMBL11702737 1.00 PTGS1 (0.63) PTGS1HPGDALDH1A1CYP2C9LMNA
Cliprofen SCHEMBL29910028 1.00 PTGS1 (0.63) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11706148 0.86 HPGD (0.46) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11703127 0.85 PTGS1 (0.68) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11703120 0.85 PTGS1 (0.68) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11703609 0.85 SMN1; SMN2 (0.46) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11702059 0.84 HPGD (0.50) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11707683 0.81 HPGD (0.42) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11707677 0.81 HPGD (0.42) PTGS1HPGDALDH1A1CYP2C9LMNA
SCHEMBL11727367 0.81 GAA (0.44) PTGS1HPGDALDH1A1CYP2C9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2838 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4335413-A2 PROSTHETIC TISSUE VALVES Cormatrix Cardiovascular, Inc. (US) 2024-03-13 EP claimed
WO-2023212179-A2 THERAPEUTIC COMPOSITIONS FOR SKIN DISORDERS AND WOUND REPAIR UNIVERSITY OF MIAMI (US) 2023-11-02 WO claimed
US-20220110979-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC 2022-04-14 US claimed
EP-3908297-A1 FIBROBLAST REGENERATIVE CELLS Figene, LLC (US) 2021-11-17 EP claimed
EP-3279663-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2021-07-28 EP claimed
WO-2020146874-A1 FIBROBLAST REGENERATIVE CELLS FIGENE, LLC (US) 2020-07-16 WO claimed
EP-3279663-A1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES The Brigham and Women's Hospital, Inc. (US) 2018-02-07 EP claimed
US-20170281724-A9 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2017-10-05 US claimed
EP-2001496-B1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES BRIGHAM & WOMENS HOSPITAL INC (US) 2017-05-31 EP claimed
US-20160228505-A1 USE OF GELSOLIN TO DIAGNOSE AND TREAT INFLAMMATORY DISEASES THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2016-08-11 US claimed
CN-1284863-A Topical compositions for NSAI drug delivery NEXMED HOLDINGS INC (US) 2001-02-21 CN claimed
EP-1003501-A4 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM & WOMENS HOSPITAL (US) 2001-01-17 EP claimed
EP-1028710-A1 TOPICAL COMPOSITIONS FOR NSAI DRUG DELIVERY Nexmed Holdings, Inc. (US) 2000-08-23 EP claimed
US-6083996-A COMPRISES ONE OR MORE NON-STEROID ANTIINFLAMMATORY AGENT, A NON-BASIC POLYMERIC SKIN PENETRATION ENHANCER AND A LIPOPHILIC SOLVENT CONTAINING ALIPHATIC ALCOHOL AND ALIPHATIC ESTER MIXTURE NEXMED HOLDINGS, INC. (US) 2000-07-04 US claimed
EP-1003501-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2000-05-31 EP claimed
WO-1999022716-A1 TOPICAL COMPOSITIONS FOR NSAI DRUG DELIVERY NEXMED HOLDINGS, INC. (US) 1999-05-14 WO claimed
WO-1998043630-A1 MEANS OF ASCERTAINING AN INDIVIDUAL'S RISK PROFILE FOR ATHEROSCLEROTIC DISEASE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 1998-10-08 WO claimed
EP-0466650-A2 Improvements in non-steroidal anti-inflammatory therapy WARNER-LAMBERT COMPANY (US) 1992-01-15 EP claimed
US-4185100-A CORTICOSTEROID AND A HYDROTROPIC ACID DERIVATIVE, ENZYME INHIBITORS JOHNSON & JOHNSON (US) 1980-01-22 US claimed
US-4035376-A ESTERS, AMIDES, HYDROXAMIC ACIDS, ANTIINFLAMMATORY JANSSEN PHARMACEUTICA N.V. (BE) 1977-07-12 US claimed