SCHEMBL4229902

SCHEMBL4229902

CC(=O)NCC(=O)N1CC(=O)[C@@H]2C1CCN2C(=O)[C@H](CC(C)C)NC(=O)c1ccc(N(C)C)cc1

nearest known ligand 0.73

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.73
CTSS P25774 3/20 0.43
PSMB9 P28065 2/20 0.39
CCR1 P32246 1/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
KMT2A Q03164 1/20 0.37
CTSV O60911 2/20 0.35
CTSL P07711 2/20 0.35
CACNA1B Q00975 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4229906 1.00 CTSK (0.73) CTSKCTSSPSMB9CCR1ALDH1A1
SCHEMBL4037181 1.00 CTSK (0.73) CTSKCTSSPSMB9CCR1ALDH1A1
SCHEMBL5941881 1.00 CTSK (0.73) CTSKCTSSPSMB9CCR1ALDH1A1
SCHEMBL4208093 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD
SCHEMBL5941844 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD
SCHEMBL4208095 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD
SCHEMBL4208090 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD
SCHEMBL4209507 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD
SCHEMBL4209501 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD
SCHEMBL5942140 0.92 CTSK (0.71) CTSKCTSSCCR1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed