SCHEMBL423183

SCHEMBL423183

COc1cc(OC)nc(C)n1

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.61
LMNA P02545 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
L3MBTL1 Q9Y468 2/20 0.46
CYP1A2 P05177 3/20 0.45
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
RECQL P46063 1/20 0.42
POLB P06746 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 1/20 0.38
HPGD P15428 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835612 0.88 PDE2A (0.52) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL7052100 0.87 PDE2A (0.55) PDE2ALMNASMN1; SMN2CYP1A2ALDH1A1
SCHEMBL29450819 0.87 PDE2A (0.55) PDE2ALMNASMN1; SMN2CYP1A2ALDH1A1
SCHEMBL25622911 0.85 PDE2A (0.53) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL12701526 0.84 PDE2A (0.48) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL9912008 0.83 PDE2A (0.52) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL30318701 0.83 PDE2A (0.52) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL11744262 0.83 PDE2A (0.52) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL10241852 0.83 PDE2A (0.52) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2
SCHEMBL8198679 0.83 PDE2A (0.52) PDE2ALMNASMN1; SMN2L3MBTL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 212 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2725022-B1 New amides as pest control agents BAYER CROPSCIENCE AG (DE) 2017-03-29 EP claimed
EP-2488510-B1 Amides and thioamides as pest control agents BAYER IP GMBH (DE) 2017-03-29 EP claimed
EP-2350090-B1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC (CA) 2015-06-03 EP claimed
EP-2297130-B1 NEW HETEROAROMATIC AMIDES AND THIOAMIDES AS PEST CONTROL AGENTS BAYER CROPSCIENCE AG (DE) 2014-09-17 EP claimed
US-8536204-B2 Amides and thioamides as pesticides BAYER CROPSCIENCE AG (DE) 2013-09-17 US claimed
US-8263606-B2 Spiro-oxindole compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2012-09-11 US claimed
EP-2410854-A2 SUBSTITUTED 1, 4-DIOXA-8-AZASPIRO Ý4,5¨DECANES USEFUL AS FUNGICIDES AND A PROCESS FOR THE PREPARATION THEREOF Council of Scientific & Industrial Research (IN) 2012-02-01 EP claimed
EP-2350090-A2 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS Xenon Pharmaceuticals Inc. (CA) 2011-08-03 EP claimed
WO-2010109299-A2 SUBSTITUTED 1, 4-DIOXA-8-AZASPIRO [4,5] DECANES USEFUL AS FUNGICIDES AND A PROCESS FOR THE PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2010-09-30 WO claimed
US-20100137299-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-06-03 US claimed
WO-2010045251-A2 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS, INC. (CA) 2010-04-22 WO claimed
WO-2025076284-A1 COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USING THE SAME DELPHIA THERAPEUTICS, INC. (US) 2025-04-10 WO disclosed
US-11912708-B2 Macrocyclic heterocycles and uses thereof KUMQUAT BIOSCIENCES INC. (US) 2024-02-27 US disclosed
US-11912708-B2 Macrocyclic heterocycles and uses thereof KUMQUAT BIOSCIENCES INC. (US) 2024-02-27 US disclosed
US-20230382907-A1 5- AND 6-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES ENLIVEN INC. 2023-11-30 US disclosed
US-5276152-A Process for the production of 4,6-dialkoxypyrimidines LONZA LTD. (CH) 1994-01-04 US disclosed
CN-1075715-A 4, the production method of 6-dialkoxy pyrimidine LONZA AG (CH) 1993-09-01 CN disclosed
EP-0552759-A1 Process for preparation of 4,6-dialkoxypyrimidines LONZA AG (CH) 1993-07-28 EP disclosed
EP-0539427-A1 PYRIMIDINYL AND TRIAZINYL HERBICIDES AgrEvo UK Limited (GB) 1993-05-05 EP disclosed
WO-1992001677-A1 PYRIMIDINYL AND TRIAZINYL HERBICIDES SCHERING AGROCHEMICALS LIMITED (GB) 1992-02-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11912708-B2 Macrocyclic heterocycles and uses thereof HRAS, KRAS, TP53 PDE2A 3207/4885LMNA 2455/4885SMN1; SMN2 1539/4885
US-20230382907-A1 5- AND 6-AZAINDOLE COMPOUNDS FOR INHIBITION OF BCR-ABL TYROSINE KINASES ABL1, ABL2, BCR PDE2A 897/4885LMNA 3763/4885SMN1; SMN2 3904/4885
US-20100137299-A1 SPIRO-OXINDOLE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS TRPV3, TRPV1, TRPC3 PDE2A 2185/4885LMNA 1296/4885SMN1; SMN2 289/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.