SCHEMBL4232811

SCHEMBL4232811

CCOc1cc(CN2CCC(Nc3nc(OC)cc(OC)n3)CC2)cc(OCC)c1Br.COc1cc(OC)nc(NC2CCNCC2)n1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 18/20 0.45
HRH1 P35367 3/20 0.45
HTR2B P41595 2/20 0.45
ACHE P22303 2/20 0.41
BACE1 P56817 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3779146 0.94 SSTR5 (0.48) SSTR5HRH1HTR2BACHEBACE1
SCHEMBL4235821 0.91 SSTR5 (0.44) SSTR5HRH1HTR2BACHEBACE1
SCHEMBL4229267 0.90 SSTR5 (0.54) SSTR5HRH1HTR2BKCNH2
SCHEMBL4224514 0.87 SSTR5 (0.45) SSTR5HRH1HTR2BACHEBACE1
SCHEMBL4231242 0.87 SSTR5 (0.50) SSTR5HRH1HTR2BACHEBACE1
SCHEMBL4220028 0.87 SSTR5 (0.58) SSTR5HRH1HTR2BKCNH2
SCHEMBL3781057 0.85 SSTR5 (0.48) SSTR5HRH1HTR2BACHEBACE1
SCHEMBL3782763 0.84 SSTR5 (0.60) SSTR5HRH1HTR2BKCNH2
SCHEMBL4226230 0.82 EHMT2 (0.49)
SCHEMBL4234199 0.82 SSTR5 (0.54) SSTR5HRH1HTR2BKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-B1 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-07-01 EP disclosed