SCHEMBL4233205

SCHEMBL4233205

Nc1ccccc1NC(=O)c1ccc(C(CCCCN2CCOCC2)NC(=O)Nc2nccs2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASR P41180 2/20 0.46
TRPV4 Q9HBA0 1/20 0.43
CYP2D6 P10635 1/20 0.41
ADORA2A P29274 1/20 0.41
SCN1A P35498 2/20 0.38
SCN5A Q14524 2/20 0.38
SCN8A Q9UQD0 2/20 0.38
HDAC1 Q13547 8/20 0.38
ALDH1A1 P00352 2/20 0.37
HRH1 P35367 1/20 0.37
TSHR P16473 1/20 0.37
HDAC3 O15379 2/20 0.37
HDAC2 Q92769 2/20 0.37
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC10 Q969S8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4235025 0.98 CASR (0.46) CASRTRPV4CYP2D6ADORA2ASCN1A
SCHEMBL4229846 0.90 HRH1 (0.40) CASRTRPV4HDAC1ALDH1A1HRH1
SCHEMBL3829026 0.89 CYP2D6 (0.50) CASRTRPV4CYP2D6ADORA2AHDAC1
SCHEMBL4223485 0.88 MAPT (0.45) CASRCYP2D6HDAC1ALDH1A1HRH1
SCHEMBL4222628 0.87 HDAC1 (0.38) HDAC1HDAC3HDAC2HDAC4HDAC7
SCHEMBL4234586 0.87 CASR (0.43) CASRTRPV4CYP2D6ADORA2ASCN1A
SCHEMBL4229410 0.87 HRH1 (0.41) CASRCYP2D6ADORA2AHDAC1ALDH1A1
SCHEMBL4224540 0.86 EPHX2 (0.48) CASRHDAC1HDAC3HDAC2SMN1; SMN2
SCHEMBL4224157 0.85 CASR (0.43) CASRTRPV4CYP2D6ADORA2ASCN1A
SCHEMBL4233251 0.85 HDAC1 (0.39) HDAC1HDAC3HDAC2HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2133339-A1 NOVEL (2-AMINOPHENYL)PYRIDINECARBOXAMIDE DERIVATIVE HAVING UREA STRUCTURE Santen Pharmaceutical Co., Ltd (JP) 2009-12-16 EP disclosed