SCHEMBL4240777

SCHEMBL4240777

COC(=O)Oc1cc(C)c2[nH]c(C3CC3)nc2c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
PDE2A O00408 6/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PARP1 P09874 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADORA1 P30542 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK4 Q16654 1/20 0.34
NPY5R Q15761 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3960529 0.80 PARP1 (0.42) CYP2D6CYP2C9LMNATP53MAPT
SCHEMBL13906484 0.80 NPY5R (0.43) CYP2D6CYP2C9LMNATP53MAPT
SCHEMBL13907999 0.75 KMT2A (0.39) CYP2D6CYP2C9MAPTPARP1NPC1
SCHEMBL13906625 0.75 NPC1 (0.37) CYP2D6CYP2C9SMN1; SMN2ADORA1NPC1
SCHEMBL4562585 0.74 MEN1 (0.38) CYP2D6CYP2C9LMNAMAPTHTT
SCHEMBL16789768 0.73 NPC1 (0.45) LMNAMAPTADORA1NPC1RAB9A
SCHEMBL13351319 0.71 KDM4E (0.42) CYP2D6CYP2C9MAPTADORA1NPC1
SCHEMBL4565286 0.71 FASN (0.37) SMN1; SMN2NPC1
SCHEMBL1542506 0.67 MAPT (0.37) MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL3965280 0.67 PARP1 (0.41) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034028-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed