SCHEMBL4244128

SCHEMBL4244128

Cc1ccc(F)cc1C(=O)N[C@@H](Cc1ccc(OCCc2cccc(N(C)c3ccccc3)n2)cc1)C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.65
ITGA5 P08648 18/20 0.65
ITGB3 P05106 15/20 0.65
ITGAV P06756 15/20 0.65
PPARG P37231 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4068834 0.85 ITGB3 (0.88) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4070827 0.79 ITGB3 (1.00) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4243117 0.77 ITGB1 (0.78) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4070628 0.77 ITGB3 (0.79) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4070162 0.77 ITGB3 (0.88) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4074598 0.77 ITGB3 (0.88) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4070455 0.77 ITGB3 (0.81) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4064435 0.76 ITGB3 (0.83) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4073748 0.76 ITGB3 (0.83) ITGB1ITGA5ITGB3ITGAV
SCHEMBL4065838 0.76 ITGB3 (0.76) ITGB1ITGA5ITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049490-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL]-L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS Astra Zeneca AB (SE) 2009-04-22 EP claimed
WO-2007141473-A1 N-(BENZOYL)-O- [2- (PYRIDIN- 2 -YLAMINO) ETHYL] -L-TYROSINE DERIVATIVES AND RELATED COMPOUNDS AS A5B1 ANTAGONISTS FOR THE TREATMENT OF SOLID TUMORS ASTRAZENECA AB (SE) 2007-12-13 WO claimed