SCHEMBL4247261

SCHEMBL4247261

Cc1nn2c(=O)n(Cc3ccccc3)c(C(C(C)C)N(CCCN)C(=O)c3ccc(Br)cc3)cc2c1Br

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 18/20 0.53
KIF23 Q02241 1/20 0.53
MAP1LC3B Q9GZQ8 2/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C19 P33261 1/20 0.51
KCNH2 Q12809 1/20 0.51
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4247266 1.00 KIF11 (0.53) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4245148 0.95 KIF11 (0.59) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4245145 0.95 KIF11 (0.59) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
Hydrochloric Acid SCHEMBL4245170 0.95 KIF11 (0.58) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
Hydrochloric Acid SCHEMBL4245173 0.95 KIF11 (0.58) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4252548 0.93 KIF11 (0.52) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4252544 0.93 KIF11 (0.52) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4244606 0.89 KIF11 (0.56) KIF11
SCHEMBL4244612 0.89 KIF11 (0.56) KIF11
SCHEMBL4253673 0.87 KIF11 (0.52) KIF11KIF23MAP1LC3BCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035426-A1 PYRAZOLOPYRIMIDONES 4SC AG (DE) 2009-03-18 EP disclosed
WO-2007144384-A1 PYRAZOLOPYRIMIDONES 4SC AG (DE) 2007-12-21 WO disclosed