SCHEMBL4248639

SCHEMBL4248639

CC(C)CN(Cc1ccc(-c2ccccn2)cc1)C(Cc1cncs1)C(O)C(Cc1ccccc1)OC(N)=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 14/20 0.39
UGT1A1 P22309 3/20 0.37
MLNR O43193 1/20 0.37
NR1I2 O75469 1/20 0.37
SLCO2B1 O94956 1/20 0.37
ABCB11 O95342 1/20 0.37
ABCB1 P08183 1/20 0.37
CCKAR P32238 1/20 0.37
OPRK1 P41145 1/20 0.37
GHSR Q92847 1/20 0.37
SLCO1B3 Q9NPD5 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
SLCO1B1 Q9Y6L6 1/20 0.37
KCNH2 Q12809 1/20 0.37
GPR142 Q7Z601 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4395637 0.85 UGT1A1 (0.42) CYP3A4UGT1A1MLNRNR1I2SLCO2B1
SCHEMBL4396378 0.82 NR1I2 (0.36) CYP3A4UGT1A1MLNRNR1I2SLCO2B1
SCHEMBL4396376 0.81 CYP3A4 (0.35) CYP3A4UGT1A1MLNRNR1I2SLCO2B1
SCHEMBL893844 0.77 CYP3A4 (0.47) CYP3A4UGT1A1MLNRNR1I2SLCO2B1
SCHEMBL893148 0.75 CYP3A4 (0.43) CYP3A4UGT1A1MLNRNR1I2SLCO2B1
SCHEMBL893146 0.75 CYP3A4 (0.43) CYP3A4UGT1A1MLNRNR1I2SLCO2B1
SCHEMBL4253307 0.73 GPR142 (0.37) CYP3A4GPR142
SCHEMBL893846 0.72 CYP3A4 (0.59) CYP3A4
SCHEMBL14118795 0.72 CYP3A4 (0.59) CYP3A4
SCHEMBL14118793 0.72 CYP3A4 (0.59) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed