SCHEMBL4248959

SCHEMBL4248959

Cc1nn2c(=O)n(Cc3ccccc3)c([C@@H](C(C)C)N(CCCNC(=O)OC(C)(C)C)C(=O)c3ccc(C(F)(F)F)cc3)cc2c1Br

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 10/20 0.45
KIF23 Q02241 1/20 0.38
TMEM97 Q5BJF2 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
MAP1LC3B Q9GZQ8 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
KCNH2 Q12809 1/20 0.36
PDE6D O43924 3/20 0.36
BRD4 O60885 1/20 0.34
P2RY14 Q15391 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
GNRHR P30968 1/20 0.34
MC4R P32245 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4251900 0.94 KIF11 (0.46) KIF11KIF23TMEM97SIGMAR1MAP1LC3B
SCHEMBL4249023 0.94 KIF11 (0.52) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4248841 0.94 KIF11 (0.47) KIF11KIF23TMEM97SIGMAR1MAP1LC3B
SCHEMBL4249025 0.94 KIF11 (0.52) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4248271 0.93 KIF11 (0.47) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4252363 0.92 KIF11 (0.46) KIF11KIF23SIGMAR1MAP1LC3BCYP3A4
SCHEMBL4252114 0.91 KIF11 (0.53) KIF11
SCHEMBL4252111 0.91 KIF11 (0.53) KIF11
SCHEMBL4248040 0.88 KIF11 (0.47) KIF11KIF23MAP1LC3BCYP3A4CYP2C19
SCHEMBL4251488 0.87 KIF11 (0.47) KIF11TMEM97SIGMAR1MAP1LC3BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035426-A1 PYRAZOLOPYRIMIDONES 4SC AG (DE) 2009-03-18 EP disclosed
WO-2007144384-A1 PYRAZOLOPYRIMIDONES 4SC AG (DE) 2007-12-21 WO disclosed