SCHEMBL4249293

SCHEMBL4249293

NCc1cnc2ncccn12

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.47
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
PKM P14618 11/20 0.44
DYRK1A Q13627 1/20 0.39
CCNK O75909 1/20 0.37
CDK12 Q9NYV4 1/20 0.37
PDE10A Q9Y233 1/20 0.34
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
HSD17B10 Q99714 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13468980 0.81 BACE1 (0.47) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL18265820 0.81 BACE1 (0.47) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL12806215 0.78 BACE1 (0.45) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL2263088 0.78 PKM (0.42) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL1204131 0.77 PKM (0.44) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL12732690 0.77 BACE1 (0.44) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL5496430 0.74 BACE1 (0.52) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL19710672 0.73 TLR7 (0.54) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL8234519 0.72 TLR7 (0.55) BACE1DRD4DRD3PKMDYRK1A
SCHEMBL303655 0.69 BACE1 (0.52) BACE1DRD4DRD3PKMDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2103614-A1 Substituted imidazopyrimidine, imidazopyrazine and imidazopyridazine derivatives as melanocortin-4 receptor modulators Santhera Pharmaceuticals (Schweiz) AG (CH) 2009-09-23 EP disclosed