SCHEMBL4251845

SCHEMBL4251845

NC(=O)c1cc2c(C3CCNCC3)cc(F)cc2n1Cc1ccccc1.NC(=O)c1cc2c(C3CCNCC3)cc(F)cc2n1Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 3/20 0.41
PLA2G10 O15496 1/20 0.40
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
PLA2G2A P14555 2/20 0.38
CCR2 P41597 2/20 0.38
F10 P00742 3/20 0.38
KCNH2 Q12809 2/20 0.37
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR1A P08908 3/20 0.36
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 3/20 0.36
SLC6A3 Q01959 3/20 0.36
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
PARP2 Q9UGN5 1/20 0.36
PARP3 Q9Y6F1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3296727 1.00 HTR6 (0.41) HTR6PLA2G10IKBKBCHUKPLA2G2A
SCHEMBL3295270 0.86 F10 (0.47) PLA2G10IKBKBCHUKPLA2G2ACCR2
Hydrochloric Acid SCHEMBL3297425 0.85 F10 (0.46) PLA2G10IKBKBCHUKPLA2G2ACCR2
SCHEMBL3299508 0.84 F10 (0.42) HTR6PLA2G10IKBKBCHUKCCR2
SCHEMBL3297073 0.84 SLC6A2 (0.42) HTR6CCR2F10KCNH2HTR1A
SCHEMBL3296497 0.83 F10 (0.46) HTR6PLA2G10CCR2F10HTR1A
Hydrochloric Acid SCHEMBL3304349 0.83 F10 (0.41) HTR6PLA2G10IKBKBCHUKCCR2
Hydrochloric Acid SCHEMBL3297955 0.83 SLC6A2 (0.42) HTR6CCR2F10KCNH2HTR1A
Hydrochloric Acid SCHEMBL3295163 0.82 F10 (0.45) HTR6PLA2G10CCR2F10HTR1A
SCHEMBL3298934 0.80 HTR6 (0.45) HTR6PLA2G10CCR2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084131-A1 INDOLE AND BENZOFURAN 2-CARBOXAMIDE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-08-05 EP disclosed
WO-2008055808-A1 INDOLE AND BENZOFURAN 2-CARBOXAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-05-15 WO disclosed