SCHEMBL4251886

SCHEMBL4251886

CNc1ccc(N2Cc3cc(OC)ccc3C2=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59
PKM P14618 2/20 0.59
POLB P06746 9/20 0.45
TP53 P04637 3/20 0.43
TDP1 Q9NUW8 4/20 0.43
MAPT P10636 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ESR1 P03372 1/20 0.43
NR4A1 P22736 1/20 0.43
APEX1 P27695 1/20 0.43
PTPN7 P35236 1/20 0.43
RECQL P46063 1/20 0.43
BLM P54132 1/20 0.43
MCL1 Q07820 1/20 0.43
ESR2 Q92731 1/20 0.43
HSD17B10 Q99714 1/20 0.43
F10 P00742 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
MAPK14 Q16539 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4250029 0.85 NPC1 (0.63) NPC1RAB9APKMPOLBTDP1
SCHEMBL4251106 0.83 NPC1 (0.43) NPC1RAB9APKMAPP
SCHEMBL4260430 0.82 APP (0.43) NPC1RAB9APKMAPP
SCHEMBL10085802 0.82 NPC1 (0.59) NPC1RAB9APKMPOLBTP53
SCHEMBL4254589 0.82 NPC1 (0.59) NPC1RAB9APKMPOLBTDP1
SCHEMBL4257367 0.81 NPC1 (0.44) NPC1RAB9APKMTP53KDM4E
SCHEMBL17541801 0.81 NPC1 (0.58) NPC1RAB9APKMPOLBMAPT
SCHEMBL4251148 0.81 NPC1 (0.58) NPC1RAB9APKMPOLBTDP1
SCHEMBL29312809 0.80 NPC1 (0.57) NPC1RAB9APKMPOLBTDP1
SCHEMBL10085457 0.77 TP53 (0.67) NPC1RAB9APKMPOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed