SCHEMBL4254589

SCHEMBL4254589

COc1ccc2c(c1)CN(c1ccc(N(C)C)cc1)C2=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.59
RAB9A P51151 5/20 0.59
PKM P14618 2/20 0.59
MAOB P27338 2/20 0.51
MAOA P21397 1/20 0.51
POLB P06746 2/20 0.45
PARP1 P09874 1/20 0.44
MELK Q14680 1/20 0.43
KDM4E B2RXH2 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
ESR1 P03372 1/20 0.43
NR4A1 P22736 1/20 0.43
APEX1 P27695 1/20 0.43
PTPN7 P35236 1/20 0.43
RECQL P46063 1/20 0.43
BLM P54132 1/20 0.43
MCL1 Q07820 1/20 0.43
ESR2 Q92731 1/20 0.43
HSD17B10 Q99714 1/20 0.43
F10 P00742 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4250029 0.85 NPC1 (0.63) NPC1RAB9APKMPOLBMELK
SCHEMBL4251146 0.83 APP (0.45) NPC1RAB9APKMMAOBMAOA
SCHEMBL4254603 0.83 NPC1 (0.51) NPC1RAB9APKMMAOBMAOA
SCHEMBL4250783 0.82 NPC1 (0.56) NPC1RAB9APKMPARP1KDM4E
SCHEMBL4254816 0.82 NPC1 (0.43) NPC1RAB9APKMPARP1HTR2C
SCHEMBL10085802 0.82 NPC1 (0.59) NPC1RAB9APKMPOLBMELK
SCHEMBL4251886 0.82 NPC1 (0.59) NPC1RAB9APKMPOLBMELK
SCHEMBL4255757 0.81 PARP1 (0.49) NPC1RAB9APKMMAOBMAOA
SCHEMBL17541801 0.81 NPC1 (0.58) NPC1RAB9APKMMAOBPOLB
SCHEMBL4258064 0.81 PARP1 (0.46) NPC1RAB9APKMPARP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO claimed
WO-2009054653-A2 ISOINDOLONES WITH HIGH BINDING AFFINITY TO BETA-AMYLOID AGGREGATES AND FIBRILS, AND ITS USE AND PREPARATION METHOD KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2009-04-30 WO disclosed