SCHEMBL4253369

SCHEMBL4253369

[CH2]CNc1nc[nH]c1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
XDH P47989 4/20 0.51
GDA Q9Y2T3 1/20 0.50
PAX8 Q06710 3/20 0.40
ALDH1A1 P00352 3/20 0.40
LMNA P02545 2/20 0.40
TSHR P16473 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MMP9 P14780 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GAA P10253 5/20 0.35
L3MBTL1 Q9Y468 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
PARP1 P09874 1/20 0.33
MKNK1 Q9BUB5 1/20 0.32
PDPK1 O15530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2458365 0.78 XDH (0.47) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL12017486 0.77 XDH (0.55) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL562980 0.76 XDH (0.67) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL2457649 0.75 XDH (0.48) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL1776355 0.74 XDH (0.47) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL1776468 0.74 XDH (0.49) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL11036315 0.74 XDH (0.60) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL2457645 0.73 XDH (0.46) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL2454476 0.73 XDH (0.46) XDHGDAPAX8ALDH1A1LMNA
SCHEMBL1776404 0.72 XDH (0.48) XDHGDAPAX8ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010535-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120098-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed