SCHEMBL4253439

SCHEMBL4253439

CCOC(=O)C1=C(C)Nc2[nH]nc(C)c2C1c1cccs1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
MAPT P10636 3/20 0.59
KMT2A Q03164 3/20 0.59
MEN1 O00255 2/20 0.59
KDM4E B2RXH2 8/20 0.54
HPGD P15428 3/20 0.54
HSD17B10 Q99714 2/20 0.54
TSHR P16473 1/20 0.54
PKM P14618 1/20 0.54
LMNA P02545 1/20 0.53
POLB P06746 1/20 0.53
AGTR1 P30556 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
GAA P10253 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
ADORA2B P29275 3/20 0.53
ADORA3 P0DMS8 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3246994 0.85 ALDH1A1 (0.47) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL1666306 0.85 ALDH1A1 (0.74) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL3004313 0.80 ALDH1A1 (0.56) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL3248414 0.77 MAPT (0.57) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL10849548 0.77 KDM4E (0.55) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL7384754 0.76 ALDH1A1 (0.62) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL7379493 0.76 ALDH1A1 (0.65) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL10789635 0.75 KDM4E (0.58) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL11752901 0.75 ALDH1A1 (1.00) ALDH1A1MAPTKMT2AMEN1KDM4E
SCHEMBL27692194 0.74 KDM4E (0.52) ALDH1A1MAPTKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed