SCHEMBL4255342

SCHEMBL4255342

C[C@]12CC[C@H]3[C@@H](CCC4CC(=O)CC[C@@]43C)[C@@H]1CC[C@@H]2OC(=O)c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
CYP19A1 P11511 6/20 0.57
GPBAR1 Q8TDU6 3/20 0.57
SHBG P04278 3/20 0.57
NR3C1 P04150 1/20 0.57
PGR P06401 1/20 0.57
SERPINA6 P08185 1/20 0.57
NR3C2 P08235 1/20 0.57
CYP3A4 P08684 1/20 0.57
AR P10275 1/20 0.57
HSD17B10 Q99714 1/20 0.57
MGAM O43451 1/20 0.57
AKR1B10 O60218 3/20 0.57
AKR1B1 P15121 3/20 0.57
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.51
OR51E2 Q9H255 1/20 0.50
KDM4E B2RXH2 1/20 0.49
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3366936 1.00 MEN1 (0.67) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL6130933 0.87 MEN1 (0.58) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL14121739 0.86 ABCB1 (0.54) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL14121738 0.86 ABCB1 (0.54) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL6130951 0.86 MEN1 (0.55) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL6913689 0.85 MEN1 (0.72) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL23363784 0.84 MEN1 (0.73) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL10971884 0.84 MEN1 (0.73) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL4252612 0.84 MEN1 (0.73) MEN1KMT2ACYP19A1GPBAR1SHBG
SCHEMBL6942662 0.84 MEN1 (0.73) MEN1KMT2ACYP19A1GPBAR1SHBG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11479802-B2 Assays for screening activity of modulators of members of the hydroxy steroid (17-beta) dehydrogenase (HSD17B) family REGENERON PHARMACEUTICALS, INC. (US) 2022-10-25 US disclosed
EP-3610029-A1 ASSAYS FOR SCREENING ACTIVITY OF MODULATORS OF MEMBERS OF THE HYDROXYSTEROID (17-BETA) DEHYDROGENASE (HSD17B) FAMILY Regeneron Pharmaceuticals, Inc. (US) 2020-02-19 EP disclosed
WO-2018190970-A1 ASSAYS FOR SCREENING ACTIVITY OF MODULATORS OF MEMBERS OF THE HYDROXYSTEROID (17-BETA) DEHYDROGENASE (HSD17B) FAMILY REGENERON PHARMACEUTICALS, INC. (US) 2018-10-18 WO disclosed
US-20180291422-A1 Assays For Screening Activity Of Modulators Of Members Of The Hydroxysteroid (17-Beta) Dehydrogenase (HSD17B) Family REGENERON PHARMACEUTICALS, INC. 2018-10-11 US disclosed
US-20090104122-A1 DETECTION OF MEMBRANE ANDROGEN RECEPTOR (mAR) AGENTS MEDEXIS S.A. (GR) 2009-04-23 US disclosed
EP-2008099-A2 DETECTION OF MEMBRANE ANDROGEN RECEPTOR (MAR) AGENTS Medexis S.A. (GR) 2008-12-31 EP disclosed
WO-2007123682-A2 DETECTION OF MEMBRANE ANDROGEN RECEPTOR (MAR) AGENTS MEDEXIS S.A. (GR) 2007-11-01 WO disclosed